SCHEMBL900479

SCHEMBL900479

NS(=O)(=O)c1ccc2nc(-c3ccc(-c4ccc(C5CCCCC5CC(=O)O)cc4)cc3)[nH]c2c1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 7/20 0.52
DGAT1 O75907 4/20 0.50
SOAT1 P35610 2/20 0.50
SCD O00767 4/20 0.48
HDAC6 Q9UBN7 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
MMP2 P08253 1/20 0.43
MMP9 P14780 1/20 0.43
NPBWR1 P48145 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL900860 0.76 DGAT1 (0.63) DGAT1SOAT1
SCHEMBL15640487 0.72 CHEK2 (0.79) CHEK2SCDHDAC6CYP3A4CYP2D6
SCHEMBL1911538 0.69 ALDH1A1 (0.67) CHEK2SCD
SCHEMBL5680021 0.69 CHEK2 (1.00) CHEK2SCD
SCHEMBL902147 0.67 DGAT1 (0.68) DGAT1SOAT1
SCHEMBL902547 0.67 DGAT1 (0.78) DGAT1SOAT1
SCHEMBL902304 0.66 DGAT1 (0.76) DGAT1SOAT1MMP2MMP9NPBWR1
SCHEMBL10189113 0.66 DGAT1 (0.64) DGAT1SOAT1SCDNPBWR1
SCHEMBL490323 0.66 HDAC6 (0.86) CHEK2SCDHDAC6CYP3A4CYP2D6
SCHEMBL30884657 0.66 HDAC6 (0.94) CHEK2SCDHDAC6CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012044567-A2 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed