SCHEMBL9006364

SCHEMBL9006364

COc1ccccc1N1CCN(CCCOc2ccc(-c3nc4ccccc4[nH]3)cc2)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 12/20 1.00
DRD2 P14416 11/20 1.00
ACHE P22303 2/20 0.62
SLC6A2 P23975 1/20 0.61
SLC6A4 P31645 1/20 0.61
DRD4 P21917 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9006339 0.87 DRD3 (1.00) DRD3DRD2ACHEDRD4
SCHEMBL601512 0.85 DRD3 (1.00) DRD3DRD2ACHE
SCHEMBL9006356 0.84 DRD3 (1.00) DRD3DRD2ACHE
SCHEMBL9006297 0.84 DRD3 (0.89) DRD3DRD2ACHE
SCHEMBL9006337 0.83 DRD3 (1.00) DRD3DRD2ACHEDRD4
SCHEMBL9006340 0.83 DRD3 (1.00) DRD3DRD2ACHE
SCHEMBL9006359 0.83 DRD3 (0.85) DRD3DRD2ACHESLC6A2SLC6A4
SCHEMBL9006348 0.83 DRD3 (0.85) DRD3DRD2ACHE
SCHEMBL9260985 0.83 ACHE (0.89) DRD3DRD2ACHE
SCHEMBL13033483 0.82 DRD2 (0.68) DRD3DRD2ACHEDRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995030659-A1 BENZIMIDAZOLE AND IMIDAZOPYRIDINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS DOPAMINERGIC AGENTS, ESP. SELECTIVE FOR THE DOPAMINE D3 RECEPTOR WARNER-LAMBERT COMPANY (US) 1995-11-16 WO claimed
US-5486517-A Benzimidazoles and imidazopyridines as central nervous system agents WARNER-LAMBERT COMPANY (US) 1996-01-23 US disclosed
WO-1995030659-A1 BENZIMIDAZOLE AND IMIDAZOPYRIDINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS DOPAMINERGIC AGENTS, ESP. SELECTIVE FOR THE DOPAMINE D3 RECEPTOR WARNER-LAMBERT COMPANY (US) 1995-11-16 WO disclosed