SCHEMBL9006728

SCHEMBL9006728

Cn1ncnc1C1CCN(C(N)=O)C1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 3/20 0.40
PDE2A O00408 4/20 0.36
BTK Q06187 5/20 0.35
APOBEC3A P31941 1/20 0.33
APOBEC3G Q9HC16 1/20 0.33
KCNH2 Q12809 1/20 0.33
HSD11B1 P28845 3/20 0.33
SPR P35270 1/20 0.33
SCD O00767 1/20 0.33
CYP11B2 P19099 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8954979 0.82 PDE4B (0.38) PDE4BPDE2ABTKKCNH2
SCHEMBL8994812 0.77 CYP3A4 (0.41) PDE4B
SCHEMBL13006565 0.74 KCNH2 (0.41) KCNH2
SCHEMBL9006694 0.73 QDPR (0.36)
SCHEMBL23107999 0.72 ESR2 (0.33) KCNH2
SCHEMBL23108006 0.72 ESR2 (0.33) KCNH2
SCHEMBL15215227 0.68 GSK3B (0.31)
SCHEMBL14413518 0.67 HSD11B1 (0.56) PDE4BHSD11B1SPRSCD
SCHEMBL29640084 0.67 HSD11B1 (0.59) HSD11B1SPR
SCHEMBL2044316 0.67 AOC3 (0.43) PDE4BHSD11B1SPR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8188085-B2 Antifungal agents MERCK SHARP & DOHME CORP. (US) 2012-05-29 US disclosed
US-20100113439-A1 Antifungal agents MERCK & CO., INC. (US) 2010-05-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100113439-A1 Antifungal agents GMDS, GBA3, UGGT1 PDE4B 671/4885PDE2A 422/4885BTK 4160/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.