SCHEMBL9006978

SCHEMBL9006978

C#Cc1cc(-c2ccc3c(c2)OC(C)(C)CC3(C)C)ccc1C(=O)OCC

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.34
RAB9A P51151 3/20 0.34
CASP3 P42574 1/20 0.34
ATM Q13315 1/20 0.34
SENP8 Q96LD8 1/20 0.34
SENP7 Q9BQF6 1/20 0.34
SENP6 Q9GZR1 1/20 0.34
HSD17B10 Q99714 4/20 0.33
ALDH1A1 P00352 3/20 0.33
KDM4E B2RXH2 3/20 0.33
GAA P10253 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
MAPT P10636 2/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
CA14 Q9ULX7 1/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9007048 0.80 RARA (0.37) NPC1RAB9ACASP3ATMSENP8
SCHEMBL9023693 0.77 NPC1 (0.36) NPC1RAB9ACASP3ATMSENP8
SCHEMBL9007121 0.76 RARA (0.43) NPC1RAB9ACASP3ATMSENP8
SCHEMBL8866206 0.73 HDAC3 (0.41) NPC1RAB9ACASP3ATMSENP8
SCHEMBL8668859 0.73 RARA (0.37) NPC1RAB9ACASP3ATMSENP8
SCHEMBL8671303 0.73 NPC1 (0.39) NPC1RAB9ACASP3ATMSENP8
SCHEMBL9845198 0.72 ALDH1A1 (0.34) HSD17B10ALDH1A1KDM4EGAAHPGD
SCHEMBL9006975 0.72 RARB (0.47) NPC1RAB9AALDH1A1SMN1; SMN2MAPT
SCHEMBL4509081 0.71 MAPT (0.38) NPC1RAB9ACASP3SENP7GAA
SCHEMBL9425665 0.71 MAPT (0.46) NPC1RAB9AATMALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0571546-B1 CHROMAN AND THIOCHROMANS WITH PHENYLETHYNYL SUBSTITUENTS AT THE 7-POSITION HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN INC (US) 1996-10-16 EP disclosed
US-5346915-A Chromans and thiochromans with phenylethynyl substituents at the 7-position having retinold-like biological activity ALLERGAN, INC. (US) 1994-09-13 US disclosed
EP-0571546-A1 CHROMAN AND THIOCHROMANS WITH PHENYLETHYNYL SUBSTITUENTS AT THE 7-POSITION HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY. ALLERGAN INC (US) 1993-12-01 EP disclosed
WO-1992014725-A1 CHROMAN AND THIOCHROMANS WITH PHENYLETHYNYL SUBSTITUENTS AT THE 7-POSITION HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN, INC. (US) 1992-09-03 WO disclosed