SCHEMBL9008707

SCHEMBL9008707

CCN(C)C(=O)NC1CCNCC1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 4/20 0.52
GNAI3 P08754 3/20 0.47
GNAO1 P09471 3/20 0.47
GNAI1 P63096 3/20 0.47
POLB P06746 1/20 0.47
EPHX2 P34913 1/20 0.38
HTR1A P08908 2/20 0.37
DRD2 P14416 2/20 0.37
DRD3 P35462 2/20 0.37
SMYD3 Q9H7B4 3/20 0.37
KCNH2 Q12809 1/20 0.36
SIGMAR1 Q99720 2/20 0.35
HTR2A P28223 1/20 0.35
CHRM5 P08912 1/20 0.35
CHRM3 P20309 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23169461 0.81 PKM (0.50) EPHX1EPHX2
SCHEMBL1596519 0.81 EPHX1 (0.59) EPHX1GNAI3GNAO1GNAI1POLB
SCHEMBL22722016 0.77 HTR1A (0.36) POLBEPHX2HTR1ADRD2DRD3
Hydrochloric Acid SCHEMBL27679507 0.77 EPHX1 (0.50) EPHX1GNAI3GNAO1GNAI1POLB
SCHEMBL12436799 0.77 HTR1A (0.36) POLBEPHX2HTR1ADRD2DRD3
SCHEMBL1315538 0.76 EPHX1 (0.51) EPHX1EPHX2SIGMAR1CHRM5CHRM3
SCHEMBL27589350 0.76 NPC1 (0.50) EPHX1
SCHEMBL24790610 0.75 EPHX1 (0.55) EPHX1GNAI3GNAO1GNAI1POLB
SCHEMBL18950691 0.75 DRD2 (0.47) HTR1ADRD2DRD3KCNH2HTR2A
SCHEMBL18950688 0.75 DRD2 (0.47) HTR1ADRD2DRD3KCNH2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576333-A ASTHMA TREATMENT ZENECA LIMITED (GB) 1996-11-19 US disclosed
US-5559131-A ANTAGONISTS OF TACHYKININS AT THE NEUROKININ 2 RECEPTOR, ANTIASTHMA ZENECA LIMITED (GB) 1996-09-24 US disclosed
US-5559132-A ANTAGONIST OF TACHYKININS AT THE NEUROKININ 2 RECEPTOR, ANTIASTHMA ZENECA LIMITED (GB) 1996-09-24 US disclosed
EP-0667858-A1 4-CARBOXOAMIDO PIPERIDINE DERIVATIVES, INTERMEDIATES AND USE AS NEUROKININ ANTAGONISTS ZENECA LIMITED (GB) 1995-08-23 EP disclosed
WO-1994010146-A1 4-CARBOXOAMIDO PIPERIDINE DERIVATIVES, INTERMEDIATES AND USE AS NEUROKININ ANTAGONISTS ZENECA LIMITED (GB) 1994-05-11 WO disclosed