SCHEMBL9010658

SCHEMBL9010658

O=C(O)CN(CCOCCOCCN(CC(=O)O)C(Cc1ccc([N+](=O)[O-])cc1)C(=O)O)CC(=O)O

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.52
BLM P54132 1/20 0.43
PMP22 Q01453 1/20 0.43
HSD17B10 Q99714 1/20 0.43
CA1 P00915 17/20 0.42
CA2 P00918 17/20 0.42
ATM Q13315 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9136161 0.89 KCNH2 (0.49) KCNH2CA2
SCHEMBL29575593 0.75 TSHR (0.49) KCNH2CA2
SCHEMBL10494760 0.75 KCNH2 (0.49) KCNH2CA2
SCHEMBL6527472 0.73 KCNH2 (0.47) KCNH2CA2
SCHEMBL9136144 0.73 KCNH2 (0.49) KCNH2CA2
SCHEMBL7598191 0.72 SLC7A5 (0.44) BLMPMP22CA1CA2
SCHEMBL7596061 0.72 CYP1A2 (0.43) BLMPMP22CA1CA2
SCHEMBL29588115 0.72 CYP1A2 (0.43) BLMPMP22CA1CA2
SCHEMBL9122751 0.72 CYP1A2 (0.45) KCNH2BLMPMP22HSD17B10CA1
SCHEMBL9435308 0.71 TDP1 (0.39) BLMPMP22CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0279307-B2 Bifunctional chelating agents ABBOTT LAB (US) 1996-11-13 EP disclosed
US-5227474-A Complexing with radioactive metals, binding to biologically active molecules for treatment of tumors and diagnostic imaging ABBOTT LABORATORIES (US) 1993-07-13 US disclosed
US-5057302-A Stable metal complexes of a substrate having a carboxymethyl arm of a polyaminopolycarboxylate framework; medical diagnosis; immunoassay; radiology; antitumor and anticarcinogenic agents ABBOTT LABORATORIES (US) 1991-10-15 US disclosed