SCHEMBL9010774

SCHEMBL9010774

CC(C)(NC(=O)c1cc(Cl)c2ccccc2c1)C(=O)C(Cl)Br

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.43
MAPT P10636 2/20 0.34
CYP1A2 P05177 2/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
PKM P14618 1/20 0.34
CYP2C19 P33261 1/20 0.34
ALDH1A1 P00352 3/20 0.34
HPGD P15428 1/20 0.34
CXCR2 P25025 1/20 0.34
KCNJ11 Q14654 2/20 0.33
POLB P06746 1/20 0.33
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
CNR2 P34972 1/20 0.32
IMPDH2 P12268 1/20 0.32
CYP2C9 P11712 1/20 0.32
MRGPRX4 Q96LA9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8400307 0.82 CNR2 (0.35) KDM4EMAPTCYP1A2CYP3A4CYP2D6
SCHEMBL8403493 0.80 CNR2 (0.34) KDM4EMAPTCYP1A2CYP3A4CYP2D6
SCHEMBL8403929 0.77 GRN (0.44) CYP2D6MEN1KMT2A
SCHEMBL9821338 0.76 PLAU (0.39) CYP1A2CYP2C19POLBMEN1KMT2A
SCHEMBL8400113 0.76 SLC6A2 (0.48) KDM4EPKMCYP2C19ALDH1A1HPGD
SCHEMBL9010823 0.75 CYP3A4 (0.43) MAPTCYP3A4ALDH1A1POLBKMT2A
SCHEMBL8400028 0.70 HPGD (0.49) KDM4EMAPTCYP1A2PKMCYP2C19
SCHEMBL9010811 0.69 HDAC1 (0.49) MAPTCYP3A4CYP2C19ALDH1A1MEN1
SCHEMBL28217120 0.68 ALDH1A1 (0.49) KDM4EMAPTALDH1A1HPGDMEN1
SCHEMBL9011451 0.68 MEN1 (0.47) KDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5547984-A FUNGICIDES ROHM AND HAAS COMPANY (US) 1996-08-20 US disclosed
US-5529978-A FUNGICIDE ROHM AND HAAS COMPANY (US) 1996-06-25 US disclosed
US-5344978-A Fungicides ROHM AND HAAS COMPANY (US) 1994-09-06 US disclosed
US-5196046-A N-acetonyl-substituted-amides ROHM AND HAAS COMPANY (US) 1993-03-23 US disclosed
EP-0170498-B1 N-ACETONYL-SUBSTITUTED-AMIDES, COMPOSITIONS CONTAINING THEM AND THEIR USE IN COMBATING FUNGI ROHM AND HAAS COMPANY (US) 1991-09-11 EP disclosed
US-4863940-A N-acetonyl-substituted amides and phytopathogenic fungicidal use thereof ROHM AND HAAS (US) 1989-09-05 US disclosed
EP-0170498-A2 N-acetonyl-substituted-amides, compositions containing them and their use in combating fungi ROHM AND HAAS COMPANY (US) 1986-02-05 EP disclosed