SCHEMBL9010823

SCHEMBL9010823

Cc1cc(C(=O)NC(C)(C)C(=O)C(Cl)Br)cc(C)n1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.43
MAPT P10636 2/20 0.36
CNR2 P34972 2/20 0.32
GRM5 P41594 1/20 0.31
POLB P06746 1/20 0.31
ALDH1A1 P00352 1/20 0.31
PRKAB2 O43741 1/20 0.31
PRKAG1 P54619 1/20 0.31
PRKAA2 P54646 1/20 0.31
PRKAA1 Q13131 1/20 0.31
PRKAG3 Q9UGI9 1/20 0.31
PRKAG2 Q9UGJ0 1/20 0.31
PRKAB1 Q9Y478 1/20 0.31
KMT2A Q03164 1/20 0.31
SCN9A Q15858 1/20 0.30
TAAR1 Q96RJ0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8403493 0.82 CNR2 (0.34) CYP3A4MAPTCNR2POLBALDH1A1
SCHEMBL8403929 0.82 GRN (0.44) KMT2A
SCHEMBL8400307 0.81 CNR2 (0.35) CYP3A4MAPTCNR2POLBALDH1A1
SCHEMBL9821338 0.75 PLAU (0.39) CNR2POLBKMT2A
SCHEMBL9821367 0.75 CNR2 (0.34) CYP3A4MAPTCNR2ALDH1A1
SCHEMBL9010774 0.75 KDM4E (0.43) CYP3A4MAPTCNR2POLBALDH1A1
SCHEMBL8400113 0.74 SLC6A2 (0.48) POLBALDH1A1KMT2A
SCHEMBL9010811 0.73 HDAC1 (0.49) CYP3A4MAPTALDH1A1KMT2A
SCHEMBL8400032 0.71 GRN (0.46) KMT2A
SCHEMBL8402033 0.69 LMNA (0.35) CYP3A4POLBALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0170498-B1 N-ACETONYL-SUBSTITUTED-AMIDES, COMPOSITIONS CONTAINING THEM AND THEIR USE IN COMBATING FUNGI ROHM AND HAAS COMPANY (US) 1991-09-11 EP claimed
EP-0170498-A2 N-acetonyl-substituted-amides, compositions containing them and their use in combating fungi ROHM AND HAAS COMPANY (US) 1986-02-05 EP claimed
US-5547984-A FUNGICIDES ROHM AND HAAS COMPANY (US) 1996-08-20 US disclosed
US-5529978-A FUNGICIDE ROHM AND HAAS COMPANY (US) 1996-06-25 US disclosed
US-5344978-A Fungicides ROHM AND HAAS COMPANY (US) 1994-09-06 US disclosed
US-5196046-A N-acetonyl-substituted-amides ROHM AND HAAS COMPANY (US) 1993-03-23 US disclosed
EP-0170498-B1 N-ACETONYL-SUBSTITUTED-AMIDES, COMPOSITIONS CONTAINING THEM AND THEIR USE IN COMBATING FUNGI ROHM AND HAAS COMPANY (US) 1991-09-11 EP disclosed
US-4863940-A N-acetonyl-substituted amides and phytopathogenic fungicidal use thereof ROHM AND HAAS (US) 1989-09-05 US disclosed
EP-0170498-A2 N-acetonyl-substituted-amides, compositions containing them and their use in combating fungi ROHM AND HAAS COMPANY (US) 1986-02-05 EP disclosed