SCHEMBL901316

SCHEMBL901316

N#Cc1cccc(-c2cccc(N)n2)c1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ASIC3 Q9UHC3 1/20 0.56
XDH P47989 1/20 0.56
IDO1 P14902 2/20 0.51
ADORA2A P29274 2/20 0.51
ADORA1 P30542 1/20 0.51
CLK4 Q9HAZ1 1/20 0.50
CDC7 O00311 1/20 0.48
CDK2 P24941 1/20 0.48
CTSS P25774 1/20 0.48
CTSK P43235 1/20 0.48
ATR Q13535 1/20 0.47
GRM5 P41594 2/20 0.47
KDM1A O60341 1/20 0.46
MAP4K4 O95819 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10431256 0.82 GABRA1 (0.59) XDHIDO1ADORA2AADORA1CLK4
SCHEMBL18105512 0.82 ASIC3 (0.60) ASIC3ADORA2ACDC7CDK2
SCHEMBL20416722 0.81 XDH (0.55) XDHIDO1ADORA2AADORA1CLK4
SCHEMBL31186635 0.81 XDH (0.55) XDHIDO1ADORA2AADORA1CLK4
SCHEMBL9792980 0.81 CTSS (0.62) XDHIDO1ADORA2AADORA1CLK4
SCHEMBL20417087 0.80 XDH (0.53) XDHIDO1ADORA2AADORA1CLK4
SCHEMBL3266995 0.79 IDO1 (0.51) XDHIDO1ADORA2ACLK4CTSS
SCHEMBL23662309 0.79 ADORA2A (0.57) XDHIDO1ADORA2AADORA1CLK4
SCHEMBL20632489 0.78 XDH (0.51) XDHIDO1ADORA2AADORA1CLK4
SCHEMBL19471325 0.77 XDH (0.65) XDHIDO1ADORA2AADORA1CLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2441755-A1 Pyridine- and isoquinoline-derivatives as Syk and JAK kinase inhibitors Almirall, S.A. (ES) 2012-04-18 EP disclosed
EP-2441755-A1 Pyridine- and isoquinoline-derivatives as Syk and JAK kinase inhibitors Almirall, S.A. (ES) 2012-04-18 EP disclosed
WO-2012041476-A1 PYRIDINE AND ISOQUINOLINE DERIVATIVES AS SYK- AND JAK-KINASE INHIBITORS ALMIRALL, S.A. (ES) 2012-04-05 WO disclosed
WO-2012041476-A1 PYRIDINE AND ISOQUINOLINE DERIVATIVES AS SYK- AND JAK-KINASE INHIBITORS ALMIRALL, S.A. (ES) 2012-04-05 WO disclosed
WO-2011136483-A1 NOVEL COMPOUNDS FOR ORGANIC ELECTRONIC MATERIAL AND ORGANIC ELECTROLUMINESCENT DEVICE USING THE SAME ROHM AND HAAS ELECTRONIC MATERIALS KOREA LTD. (KR) 2011-11-03 WO disclosed