SCHEMBL9013352

SCHEMBL9013352

COc1ccc(-c2nc(OCCN3CCN(C(c4ccccc4)c4ccccc4)CC3)cc(C(F)(F)F)n2)cc1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
TDP1 Q9NUW8 1/20 0.46
ESR1 P03372 2/20 0.46
CACNA1A O00555 1/20 0.43
CACNA2D1 P54289 1/20 0.43
CACNB1 Q02641 1/20 0.43
ALOX5 P09917 1/20 0.43
ALDH1A1 P00352 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALOX15 P16050 1/20 0.41
LMNA P02545 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
MAPK1 P28482 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9013419 0.92 ESR1 (0.45) MEN1KMT2AESR1ALOX5ALDH1A1
SCHEMBL9013654 0.92 KMT2A (0.50) MEN1KMT2ATDP1ALOX5ALDH1A1
SCHEMBL9013760 0.90 CYP2D6 (0.48) MEN1KMT2ATDP1CACNA1ACACNA2D1
SCHEMBL9013334 0.90 KMT2A (0.49) MEN1KMT2ATDP1ALOX5ALDH1A1
SCHEMBL9013604 0.88 MEN1 (0.52) MEN1KMT2ATDP1ESR1ALOX5
SCHEMBL9013385 0.86 MEN1 (0.47) MEN1KMT2ATDP1
SCHEMBL9013689 0.85 ACHE (0.47) MEN1KMT2ATDP1ALOX5
SCHEMBL9013518 0.83 CYP2D6 (0.46) MEN1KMT2AALOX5
SCHEMBL9013570 0.81 ACHE (0.44) MEN1KMT2AALOX5
SCHEMBL9013417 0.81 ESR1 (0.46) MEN1KMT2AESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5589477-A LEARNING ENHANCEMENT, CNS NIPPON SHINYAKU COMPANY, LIMITED (JP) 1996-12-31 US disclosed
EP-0555478-A1 PYRIMIDINE DERIVATIVE AND MEDICINE NIPPON SHINYAKU COMPANY, LIMITED (JP) 1993-08-18 EP disclosed