SCHEMBL9013760

SCHEMBL9013760

FC(F)(F)c1ccc(-c2nc(OCCN3CCN(C(c4ccccc4)c4ccccc4)CC3)cc(C(F)(F)F)n2)cc1

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.48
KMT2A Q03164 2/20 0.47
MEN1 O00255 1/20 0.47
TDP1 Q9NUW8 1/20 0.46
ALOX5 P09917 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.42
ALDH1A1 P00352 2/20 0.42
MAPT P10636 2/20 0.42
MAPK1 P28482 2/20 0.42
HTT P42858 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
CACNA1A O00555 1/20 0.41
CACNA2D1 P54289 1/20 0.41
CACNA1B Q00975 1/20 0.41
CACNB1 Q02641 1/20 0.41
CACNA1C Q13936 1/20 0.41
LMNA P02545 1/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9013654 0.94 KMT2A (0.50) KMT2AMEN1TDP1ALOX5ALDH1A1
SCHEMBL9013334 0.92 KMT2A (0.49) KMT2AMEN1TDP1ALOX5ALDH1A1
SCHEMBL9013570 0.91 ACHE (0.44) CYP2D6KMT2AMEN1ALOX5
SCHEMBL9013518 0.91 CYP2D6 (0.46) CYP2D6KMT2AMEN1ALOX5
SCHEMBL9013352 0.90 MEN1 (0.52) KMT2AMEN1TDP1ALOX5L3MBTL1
SCHEMBL9013385 0.89 MEN1 (0.47) KMT2AMEN1TDP1
SCHEMBL9013689 0.87 ACHE (0.47) KMT2AMEN1TDP1ALOX5
SCHEMBL9013561 0.82 ACHE (0.44)
SCHEMBL9013419 0.81 ESR1 (0.45) KMT2AMEN1ALOX5ALDH1A1MAPT
SCHEMBL9013406 0.80

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5589477-A LEARNING ENHANCEMENT, CNS NIPPON SHINYAKU COMPANY, LIMITED (JP) 1996-12-31 US disclosed
EP-0555478-A1 PYRIMIDINE DERIVATIVE AND MEDICINE NIPPON SHINYAKU COMPANY, LIMITED (JP) 1993-08-18 EP disclosed