SCHEMBL9013570

SCHEMBL9013570

Fc1ccc(C(c2ccc(F)cc2)N2CCN(CCOc3cc(C(F)(F)F)nc(-c4ccc(C(F)(F)F)cc4)n3)CC2)cc1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACHE P22303 3/20 0.44
CYP2D6 P10635 1/20 0.41
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
KCNH2 Q12809 1/20 0.38
DRD2 P14416 4/20 0.38
DRD4 P21917 4/20 0.38
DRD3 P35462 4/20 0.38
ALOX5 P09917 1/20 0.38
HRH1 P35367 1/20 0.38
MC4R P32245 1/20 0.38
HTR2A P28223 1/20 0.38
HTR7 P34969 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9013689 0.96 ACHE (0.47) ACHEMEN1KMT2ADRD2DRD4
SCHEMBL9013385 0.91 MEN1 (0.47) ACHEMEN1KMT2A
SCHEMBL9013760 0.91 CYP2D6 (0.48) CYP2D6MEN1KMT2AALOX5
SCHEMBL9013334 0.91 KMT2A (0.49) ACHEMEN1KMT2ADRD2DRD4
SCHEMBL9013561 0.91 ACHE (0.44) ACHEKCNH2
SCHEMBL9013419 0.90 ESR1 (0.45) ACHEMEN1KMT2AKCNH2DRD2
SCHEMBL9013654 0.85 KMT2A (0.50) MEN1KMT2AALOX5
SCHEMBL9013518 0.82 CYP2D6 (0.46) CYP2D6MEN1KMT2AALOX5
SCHEMBL9013352 0.81 MEN1 (0.52) MEN1KMT2AALOX5
SCHEMBL9013766 0.79 MEN1 (0.47) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5589477-A LEARNING ENHANCEMENT, CNS NIPPON SHINYAKU COMPANY, LIMITED (JP) 1996-12-31 US disclosed
EP-0555478-A1 PYRIMIDINE DERIVATIVE AND MEDICINE NIPPON SHINYAKU COMPANY, LIMITED (JP) 1993-08-18 EP disclosed