SCHEMBL9014400

SCHEMBL9014400

COc1ccc(C2CCN(CCC3CCCOc4ccc(O)cc43)CC2)cc1OC

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.69
QDPR P09417 1/20 0.41
MEN1 O00255 1/20 0.40
P4HB P07237 1/20 0.40
KMT2A Q03164 1/20 0.40
DRD2 P14416 3/20 0.38
TLR9 Q9NR96 3/20 0.38
TLR7 Q9NYK1 3/20 0.38
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37
TLR4 O00206 1/20 0.37
TLR3 O15455 1/20 0.37
TLR8 Q9NR97 1/20 0.37
DRD3 P35462 3/20 0.37
ALDH1A1 P00352 2/20 0.37
CYP1A2 P05177 2/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2D6 P10635 2/20 0.37
CYP2C19 P33261 2/20 0.37
OPRM1 P35372 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9014779 0.90 KCNH2 (0.70) KCNH2DRD2DRD4
SCHEMBL9014758 0.89 KCNH2 (0.69) KCNH2QDPRDRD2TLR9TLR7
SCHEMBL9014729 0.89 KCNH2 (0.69) KCNH2QDPRMEN1KMT2ADRD2
SCHEMBL9014359 0.88 KCNH2 (0.89) KCNH2DRD2TLR9TLR7
SCHEMBL9014376 0.86 KCNH2 (0.66) KCNH2DRD2TLR9TLR7TLR4
SCHEMBL9677908 0.83 KCNH2 (0.77) KCNH2QDPRDRD2TLR9TLR7
Hydrochloric Acid SCHEMBL10407809 0.82 KCNH2 (0.76) KCNH2DRD2TLR9TLR7TLR4
Terikalant SCHEMBL1815992 0.82 KCNH2 (1.00) KCNH2QDPRDRD2TLR9TLR7
Terikalant SCHEMBL30770792 0.82 KCNH2 (1.00) KCNH2QDPRDRD2TLR9TLR7
Terikalant SCHEMBL9678648 0.82 KCNH2 (1.00) KCNH2QDPRDRD2TLR9TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5495022-A Piperidines and piperazines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-02-27 US disclosed
EP-0634398-A1 4-Phenylpiperidinyl-1/-piperazinyl-1-ethylsubstituted benzofusedheterocycles as antiarrhythmic agents MERCK PATENT GmbH (DE) 1995-01-18 EP disclosed