SCHEMBL9014729

SCHEMBL9014729

COc1ccc(C2CCN(CCC3CCCOc4ccc(Cl)cc43)CC2)cc1OC

nearest known ligand 0.69

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.69
TLR9 Q9NR96 5/20 0.42
TLR7 Q9NYK1 5/20 0.42
DRD2 P14416 2/20 0.39
CCR2 P41597 1/20 0.38
TLR4 O00206 1/20 0.37
TLR3 O15455 1/20 0.37
TLR8 Q9NR97 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
ALDH1A1 P00352 1/20 0.37
QDPR P09417 1/20 0.36
DRD4 P21917 1/20 0.36
MAPK1 P28482 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
SIGMAR1 Q99720 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9014779 0.90 KCNH2 (0.70) KCNH2DRD2DRD4SIGMAR1
SCHEMBL9014758 0.89 KCNH2 (0.69) KCNH2TLR9TLR7DRD2TLR4
SCHEMBL9014400 0.89 KCNH2 (0.69) KCNH2TLR9TLR7DRD2TLR4
SCHEMBL9014359 0.88 KCNH2 (0.89) KCNH2TLR9TLR7DRD2SIGMAR1
SCHEMBL9014376 0.86 KCNH2 (0.66) KCNH2TLR9TLR7DRD2TLR4
SCHEMBL9677908 0.83 KCNH2 (0.77) KCNH2TLR9TLR7DRD2TLR4
SCHEMBL9015278 0.83 KCNH2 (0.65) KCNH2TLR9TLR7DRD2TLR4
Hydrochloric Acid SCHEMBL10407809 0.82 KCNH2 (0.76) KCNH2TLR9TLR7DRD2TLR4
Terikalant SCHEMBL30770792 0.82 KCNH2 (1.00) KCNH2TLR9TLR7DRD2TLR4
Terikalant SCHEMBL1815992 0.82 KCNH2 (1.00) KCNH2TLR9TLR7DRD2TLR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5495022-A Piperidines and piperazines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-02-27 US disclosed
EP-0634398-A1 4-Phenylpiperidinyl-1/-piperazinyl-1-ethylsubstituted benzofusedheterocycles as antiarrhythmic agents MERCK PATENT GmbH (DE) 1995-01-18 EP disclosed