SCHEMBL9014725

SCHEMBL9014725

COc1ccc(C2CCN(CCC3CCN(C(C)=O)c4ccccc43)CC2)cc1OC

nearest known ligand 0.63

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.63
PDE4B Q07343 4/20 0.46
PDE4A P27815 2/20 0.46
PDE4C Q08493 2/20 0.46
PDE4D Q08499 2/20 0.46
QDPR P09417 2/20 0.44
DRD2 P14416 4/20 0.44
HTR1A P08908 1/20 0.42
HTR2A P28223 1/20 0.42
CCR5 P51681 2/20 0.40
SLC18A3 Q16572 1/20 0.40
TRIM24 O15164 1/20 0.40
BRPF1 P55201 1/20 0.40
HTR2C P28335 1/20 0.40
DRD4 P21917 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9014708 0.91 KCNH2 (0.61) KCNH2PDE4BPDE4APDE4CPDE4D
SCHEMBL9014839 0.87 DRD2 (0.54) KCNH2DRD2HTR1AHTR2ASLC18A3
SCHEMBL9014370 0.86 KCNH2 (0.70) KCNH2PDE4BPDE4APDE4CPDE4D
SCHEMBL9014780 0.83 KCNH2 (0.66) KCNH2QDPRDRD2HTR2C
SCHEMBL9014652 0.83 KCNH2 (0.48) KCNH2DRD2HTR1AHTR2ACCR5
SCHEMBL9014362 0.82 KCNH2 (0.65) KCNH2QDPRDRD2HTR2C
SCHEMBL9014375 0.80 KCNH2 (0.70) KCNH2PDE4BPDE4APDE4CPDE4D
SCHEMBL9014688 0.78 KCNH2 (0.67) KCNH2DRD2DRD4
SCHEMBL6792592 0.78 DRD2 (0.52) KCNH2DRD2HTR1AHTR2ASLC18A3
SCHEMBL9014672 0.78 DRD2 (0.55) KCNH2DRD2SLC18A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5495022-A Piperidines and piperazines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-02-27 US disclosed
EP-0634398-A1 4-Phenylpiperidinyl-1/-piperazinyl-1-ethylsubstituted benzofusedheterocycles as antiarrhythmic agents MERCK PATENT GmbH (DE) 1995-01-18 EP disclosed