SCHEMBL9014839

SCHEMBL9014839

COc1ccc(C2CCN(CCC3CCN(C(C)=O)c4ccccc43)CC2)cc1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 4/20 0.54
OPRM1 P35372 1/20 0.48
BRD4 O60885 1/20 0.47
BRD2 P25440 1/20 0.47
BRD3 Q15059 1/20 0.47
KCNH2 Q12809 2/20 0.46
SIGMAR1 Q99720 2/20 0.45
SLC18A3 Q16572 1/20 0.45
HTR1A P08908 1/20 0.44
HTR2A P28223 1/20 0.44
CHRM4 P08173 1/20 0.44
HSD11B1 P28845 1/20 0.41
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
CCR2 P41597 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9014672 0.90 DRD2 (0.55) DRD2OPRM1KCNH2SIGMAR1SLC18A3
SCHEMBL9014725 0.87 KCNH2 (0.63) DRD2KCNH2SLC18A3HTR1AHTR2A
SCHEMBL9014679 0.82 DRD2 (0.57) DRD2OPRM1KCNH2SIGMAR1CHRM4
SCHEMBL11839176 0.82 DRD2 (0.57) DRD2OPRM1SIGMAR1SLC18A3HTR1A
SCHEMBL6790341 0.81 DRD2 (0.55) DRD2OPRM1KCNH2SIGMAR1SLC18A3
SCHEMBL9014652 0.81 KCNH2 (0.48) DRD2KCNH2HTR1AHTR2A
SCHEMBL9014749 0.79 DRD2 (0.53) DRD2OPRM1SIGMAR1SLC18A3
SCHEMBL28752384 0.79 DRD2 (0.55) DRD2OPRM1KCNH2SIGMAR1SLC18A3
SCHEMBL11823970 0.78 DRD2 (0.52) DRD2SLC18A3HTR1AHTR2ACCR2
SCHEMBL9014708 0.78 KCNH2 (0.61) DRD2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5495022-A Piperidines and piperazines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-02-27 US disclosed
EP-0634398-A1 4-Phenylpiperidinyl-1/-piperazinyl-1-ethylsubstituted benzofusedheterocycles as antiarrhythmic agents MERCK PATENT GmbH (DE) 1995-01-18 EP disclosed