SCHEMBL9014652

SCHEMBL9014652

CC(=O)N1CCC(CCN2CCC(c3ccc4c(c3)OCO4)CC2)c2ccccc21

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.48
DRD2 P14416 11/20 0.43
HTR2A P28223 10/20 0.43
DRD3 P35462 9/20 0.43
SCN9A Q15858 1/20 0.43
HTR1A P08908 1/20 0.42
SLC6A4 P31645 1/20 0.42
CCR5 P51681 1/20 0.42
HTT P42858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9014782 0.91 KCNH2 (0.47) KCNH2DRD2HTR2ADRD3SCN9A
SCHEMBL9014725 0.83 KCNH2 (0.63) KCNH2DRD2HTR2AHTR1ACCR5
SCHEMBL9014765 0.82 KCNH2 (0.50) KCNH2DRD2HTR2ADRD3SCN9A
SCHEMBL9014839 0.81 DRD2 (0.54) KCNH2DRD2HTR2AHTR1A
SCHEMBL11833053 0.79 SLC18A3 (0.45) KCNH2DRD2HTR2ADRD3HTR1A
SCHEMBL6792592 0.78 DRD2 (0.52) KCNH2DRD2HTR2AHTR1ASLC6A4
SCHEMBL11839176 0.77 DRD2 (0.57) DRD2HTR2AHTR1A
SCHEMBL6790341 0.77 DRD2 (0.55) KCNH2DRD2HTR2ADRD3HTR1A
SCHEMBL28752384 0.74 DRD2 (0.55) KCNH2DRD2HTR2AHTR1A
SCHEMBL9014749 0.74 DRD2 (0.53) DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5495022-A Piperidines and piperazines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-02-27 US disclosed
EP-0634398-A1 4-Phenylpiperidinyl-1/-piperazinyl-1-ethylsubstituted benzofusedheterocycles as antiarrhythmic agents MERCK PATENT GmbH (DE) 1995-01-18 EP disclosed