SCHEMBL9014858

SCHEMBL9014858

c1ccc(N2CCN(CCCCCOc3cnc4c(n3)CCCC4)CC2)nc1

nearest known ligand 0.63

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.57
HRH3 Q9Y5N1 4/20 0.53
DRD2 P14416 6/20 0.52
HTR1A P08908 5/20 0.52
HTR2A P28223 5/20 0.52
HTR7 P34969 5/20 0.52
DRD3 P35462 4/20 0.52
DRD1 P21728 3/20 0.52
DRD4 P21917 2/20 0.52
ADRA2C P18825 2/20 0.52
DRD5 P21918 2/20 0.52
HRH1 P35367 2/20 0.52
POLB P06746 1/20 0.51
MAOB P27338 4/20 0.50
MAOA P21397 2/20 0.50
HTR6 P50406 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9014815 0.99 KCNH2 (0.55) KCNH2HRH3DRD2HTR1AHTR2A
SCHEMBL9014685 0.96 DRD3 (0.57) KCNH2HRH3DRD2HTR1AHTR2A
SCHEMBL9014901 0.92 SLC6A2 (0.58) KCNH2HRH3DRD2HTR1AHTR2A
SCHEMBL9014904 0.86 HRH3 (0.49) KCNH2HRH3DRD2HTR1AHTR2A
SCHEMBL9014893 0.85 HRH3 (0.50) KCNH2HRH3DRD2HTR1AHTR2A
SCHEMBL9014870 0.84 HTR3E (0.45) KCNH2DRD2HTR1AHTR2AHTR7
SCHEMBL9014892 0.84 KCNH2 (0.56) KCNH2HRH3DRD2HTR1AHTR2A
SCHEMBL9014817 0.83 HTR1A (0.52) KCNH2HRH3DRD2HTR1AHTR2A
SCHEMBL9265535 0.83 KDM4E (0.44) KCNH2HRH3DRD2HTR1AHTR2A
SCHEMBL9180538 0.82 HRH3 (0.58) KCNH2HRH3DRD2HTR1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5578596-A TREATMENT OF SEROTONERGIC NEURON RELATED DISEASES, MOTION SICKNESS, ANXIXETY, DEPRESSION ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1996-11-26 US disclosed
EP-0668276-A1 2-ALKOXY-5,6,7,8-TETRAHYDROQUINOXALINE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1995-08-23 EP disclosed