SCHEMBL9014893

SCHEMBL9014893

c1cnc(N2CCN(CCCCOc3cnc4c(n3)CCCC4)CC2)nc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 5/20 0.50
DRD2 P14416 5/20 0.49
DRD3 P35462 5/20 0.49
HTR1A P08908 5/20 0.48
HTR2A P28223 3/20 0.48
DRD1 P21728 2/20 0.48
DRD5 P21918 1/20 0.48
ALDH1A1 P00352 2/20 0.47
SLC22A2 O15244 1/20 0.47
ABCB11 O95342 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
ADRA2C P18825 1/20 0.47
CNR1 P21554 1/20 0.47
ADRA1D P25100 1/20 0.47
HTR2C P28335 1/20 0.47
HTR7 P34969 1/20 0.47
ADRA1A P35348 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9014904 0.99 HRH3 (0.49) HRH3DRD2DRD3HTR1AHTR2A
SCHEMBL9014894 0.96 DRD2 (0.52) HRH3DRD2DRD3HTR1AHTR2A
SCHEMBL9014695 0.93 SLC6A2 (0.45) HRH3DRD2DRD3HTR1AHTR2A
SCHEMBL9014823 0.87 HRH3 (0.43) HRH3DRD2DRD3HTR1AHTR2A
SCHEMBL9014815 0.86 KCNH2 (0.55) HRH3DRD2DRD3HTR1AHTR2A
SCHEMBL9014676 0.86 HTR1A (0.47) HRH3DRD3HTR1AKCNH2
SCHEMBL9014858 0.85 KCNH2 (0.57) HRH3DRD2DRD3HTR1AHTR2A
SCHEMBL9014715 0.85 HTR1A (0.43) HTR1A
SCHEMBL9014886 0.83 DRD3 (0.46) HRH3DRD2DRD3HTR1AHTR2A
SCHEMBL9014685 0.82 DRD3 (0.57) HRH3DRD2DRD3HTR1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5578596-A TREATMENT OF SEROTONERGIC NEURON RELATED DISEASES, MOTION SICKNESS, ANXIXETY, DEPRESSION ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1996-11-26 US disclosed
EP-0668276-A1 2-ALKOXY-5,6,7,8-TETRAHYDROQUINOXALINE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1995-08-23 EP disclosed