SCHEMBL9014929

SCHEMBL9014929

C[Si](C)(C)C#Cc1cccc(Sc2cccc(F)c2C#N)c1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AR P10275 4/20 0.36
PGR P06401 1/20 0.36
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
HSD17B10 Q99714 1/20 0.32
L3MBTL1 Q9Y468 2/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
GRM5 P41594 1/20 0.30
MAOA P21397 1/20 0.30
MAOB P27338 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1154616 0.77 L3MBTL1 (0.44) ARPGRKDM4EALDH1A1HPGD
SCHEMBL9082431 0.76 MEN1 (0.36) ALDH1A1MEN1KMT2ANPSR1GRM5
SCHEMBL9015004 0.74 AR (0.42) ARPGRKDM4EALDH1A1HPGD
SCHEMBL8410613 0.74 DHFR (0.44) ARPGRKDM4EALDH1A1HPGD
SCHEMBL8410372 0.73 AR (0.40) ARPGRKDM4EALDH1A1HPGD
SCHEMBL2075358 0.71 L3MBTL1 (0.42) ARPGRKDM4EALDH1A1HPGD
SCHEMBL9014961 0.71 GRM5 (0.39) GRM5
SCHEMBL2768310 0.70 GRM5 (0.36) KDM4EALDH1A1HPGDHSD17B10MEN1
SCHEMBL853825 0.70 GRM5 (0.49) GRM5
SCHEMBL19781320 0.68 TRPV4 (0.45) GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0746542-A1 THERAPEUTIC BENZONITRILES THE WELLCOME FOUNDATION LIMITED (GB) 1996-12-11 EP disclosed
WO-1995023134-A1 THERAPEUTIC BENZONITRILES THE WELLCOME FOUNDATION LIMITED (GB) 1995-08-31 WO disclosed