SCHEMBL9015308

SCHEMBL9015308

Brc1ccc2c(c1)CCCC2CCN1CCN(c2ccc3c(c2)OCCO3)CC1

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 4/20 0.45
DRD3 P35462 3/20 0.45
SIGMAR1 Q99720 2/20 0.45
HTR1A P08908 2/20 0.45
ADRA2A P08913 1/20 0.45
ADRA2C P18825 1/20 0.45
ADRA1D P25100 1/20 0.45
ADRA1A P35348 1/20 0.45
ADRA1B P35368 1/20 0.45
DRD4 P21917 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9014718 0.88 DRD2 (0.45) DRD2DRD3SIGMAR1HTR1AADRA2A
SCHEMBL9014693 0.87 SIGMAR1 (0.55) DRD2DRD3SIGMAR1HTR1AADRA2A
SCHEMBL9014658 0.82 MEN1 (0.41) DRD2DRD3SIGMAR1HTR1AADRA2A
SCHEMBL7812153 0.76 HTR1A (0.63) DRD2DRD3SIGMAR1HTR1AADRA2A
Hydrochloric Acid SCHEMBL10408656 0.75 HTR1A (0.53) DRD2DRD3SIGMAR1HTR1AADRA2A
SCHEMBL6974927 0.74 DRD2 (0.49) DRD2DRD3SIGMAR1HTR1AADRA2A
SCHEMBL17226487 0.72 DRD2 (0.54) DRD2DRD3SIGMAR1HTR1AADRA2A
Hydrochloric Acid SCHEMBL10407883 0.71 KCNH2 (0.50) DRD2DRD3SIGMAR1HTR1AADRA2A
SCHEMBL9014731 0.70 MAPT (0.42) DRD2DRD3SIGMAR1HTR1AADRA2A
SCHEMBL6977453 0.70 DRD2 (0.47) DRD2DRD3SIGMAR1HTR1AADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5495022-A Piperidines and piperazines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-02-27 US disclosed
EP-0634398-A1 4-Phenylpiperidinyl-1/-piperazinyl-1-ethylsubstituted benzofusedheterocycles as antiarrhythmic agents MERCK PATENT GmbH (DE) 1995-01-18 EP disclosed