SCHEMBL9017562

SCHEMBL9017562

N#CC(C(=O)Nc1ccc(Oc2ccc(F)cc2)cc1)=C(O)C1CCCC1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 2/20 0.59
ENPP3 O14638 3/20 0.46
ENPP1 P22413 2/20 0.46
ENPP2 Q13822 2/20 0.46
EPHX2 P34913 3/20 0.45
RAB9A P51151 4/20 0.43
NPC1 O15118 3/20 0.43
EPHX1 P07099 2/20 0.42
FNTA P49354 1/20 0.42
FNTB P49356 1/20 0.42
TP53 P04637 1/20 0.41
MAPK10 P53779 1/20 0.41
ALDH1A1 P00352 2/20 0.41
MAPT P10636 1/20 0.41
CYP1A2 P05177 1/20 0.41
GAA P10253 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
GLA P06280 1/20 0.40
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9017616 0.98 DHODH (0.59) DHODHENPP3ENPP1ENPP2EPHX2
SCHEMBL9017543 0.95 DHODH (0.65) DHODHEPHX2RAB9AFNTAFNTB
SCHEMBL9310653 0.90 DHODH (0.58) DHODHEPHX2RAB9ATP53MAPK10
SCHEMBL25813258 0.88 DHODH (0.74) DHODHRAB9ANPC1EPHX1TP53
SCHEMBL27242987 0.88 DHODH (0.74) DHODHRAB9ANPC1EPHX1TP53
SCHEMBL9157076 0.85 DHODH (0.64) DHODHEPHX2RAB9ANPC1EPHX1
SCHEMBL8614830 0.84 DHODH (0.69) DHODHRAB9ANPC1TP53MAPK10
SCHEMBL9017605 0.83 DHODH (0.61) DHODHEPHX2RAB9AEPHX1FNTA
SCHEMBL9017561 0.83 DHODH (0.61) DHODHEPHX2RAB9ANPC1FNTA
SCHEMBL9017547 0.83 DHODH (0.61) DHODHEPHX2RAB9AFNTAFNTB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0533573-B1 Derivatives of 3-cyclo alkyl-propen-2-amide, their tautomeres and salts and their use as antiinflammatory agents ROUSSEL UCLAF (FR) 1996-12-04 EP disclosed
US-5389652-A Antiinflammatory agent ROUSSEL-UCLAF (FR) 1995-02-14 US disclosed
US-5312830-A Antiinflammatory agents ROUSSEL-UCLAF (FR) 1994-05-17 US disclosed
EP-0533573-A2 Derivatives of 3-cyclo alkyl-propen-2-amide, their tautomeres and salts and their use as antiinflammatory agents ROUSSEL UCLAF (FR) 1993-03-24 EP disclosed