SCHEMBL9018129

SCHEMBL9018129

CCC(CC)OC(=O)Oc1ccc(C(=O)NS(=O)(=O)c2ccc(CCNC(=O)Cc3ccccc3)cc2)cn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.46
CA2 P00918 4/20 0.46
CA5A P35218 2/20 0.46
CA7 P43166 2/20 0.46
CA5B Q9Y2D0 2/20 0.46
OPRM1 P35372 3/20 0.43
OPRD1 P41143 3/20 0.43
OPRK1 P41145 1/20 0.43
P4HTM Q9NXG6 2/20 0.41
RORC P51449 1/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
MAPT P10636 1/20 0.39
MEN1 O00255 1/20 0.39
POLB P06746 1/20 0.39
KMT2A Q03164 1/20 0.39
CA12 O43570 2/20 0.39
CA9 Q16790 2/20 0.39
ALDH1A1 P00352 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9018569 0.93 ALDH1A1 (0.43) OPRM1OPRD1OPRK1P4HTMRAB9A
SCHEMBL9018345 0.93 OPRM1 (0.40) CA1CA2CA5ACA7CA5B
SCHEMBL9018171 0.93 CA1 (0.45) CA1CA2CA5ACA7CA5B
SCHEMBL9018332 0.93 CA1 (0.45) CA1CA2CA5ACA7CA5B
SCHEMBL9018475 0.92 CA1 (0.47) CA1CA2CA5ACA7CA5B
SCHEMBL9017989 0.92 NPC1 (0.48) CA1CA2CA7OPRM1OPRD1
SCHEMBL9018302 0.92 CA1 (0.50) CA1CA2CA5ACA7CA5B
SCHEMBL9018380 0.91 MEN1 (0.46) OPRM1OPRD1OPRK1P4HTMNPC1
SCHEMBL9018484 0.90 POLB (0.49) OPRM1OPRD1OPRK1MAPTMEN1
SCHEMBL9018211 0.89 ALDH1A1 (0.46) OPRM1OPRD1OPRK1P4HTMRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0590520-B1 Acylsulphonamido and sulphonamidopyridine-2-carboxylic acid esters, pyridine-n-oxides thereof, a process for their preparation and their use as medicaments HOECHST AG (DE) 1996-06-12 EP disclosed
EP-0590520-A1 Acylsulphonamido and sulphonamidopyridine-2-carboxylic acid esters, pyridine-n-oxides thereof, a process for their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1994-04-06 EP disclosed