SCHEMBL9018716

SCHEMBL9018716

NC(N)=NC(=O)c1ccc(C(F)(F)F)cc1C(F)(F)F

nearest known ligand 0.62

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.62
ALDH1A1 P00352 3/20 0.46
KDM4E B2RXH2 1/20 0.46
HPGD P15428 1/20 0.46
HSD17B10 Q99714 1/20 0.46
SLC9A1 P19634 6/20 0.46
PLAU P00749 2/20 0.45
SLC9A5 Q14940 1/20 0.44
FLT1 P17948 1/20 0.43
FLT4 P35916 1/20 0.43
KDR P35968 1/20 0.43
CFTR P13569 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8609836 0.89 CFTR (0.57) CES2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL9018662 0.87 CES2 (0.62) CES2ALDH1A1KDM4EHPGDHSD17B10
Hydrochloric Acid SCHEMBL8393438 0.86 CES2 (0.60) CES2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL9018696 0.84 GAA (0.51) CES2ALDH1A1KDM4EHPGDHSD17B10
Hydrochloric Acid SCHEMBL8394096 0.83 SLC9A1 (0.45) CES2SLC9A1PLAUCYP3A4CYP2C19
Hydrochloric Acid SCHEMBL8393386 0.83 GAA (0.50) CES2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL1002163 0.81 CES2 (0.72) CES2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL9018707 0.81 SLC9A1 (0.46) CES2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL9018685 0.80 CES2 (0.49) CES2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL9018705 0.79 SLC9A1 (0.48) CES2SLC9A1PLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0743301-A2 Benzoylguanidines containing fluorine MERCK PATENT GmbH (DE) 1996-11-20 EP disclosed