SCHEMBL9018723

SCHEMBL9018723

CCCCc1ccc(OC(F)(F)F)cc1C(=O)N=C(N)N

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 1/20 0.40
ACR P10323 1/20 0.40
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
ALOX5 P09917 1/20 0.38
PPARG P37231 1/20 0.38
NOS3 P29474 2/20 0.36
NOS1 P29475 2/20 0.36
NOS2 P35228 2/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
NR1H2 P55055 1/20 0.35
NR1H3 Q13133 1/20 0.35
PCSK9 Q8NBP7 1/20 0.35
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8609393 0.94 HDAC3 (0.38) PRSS1ACRHDAC3HDAC1HDAC2
SCHEMBL9018706 0.93 PTGS1 (0.38) HDAC3HDAC1HDAC2NOS3NOS1
SCHEMBL9018679 0.89 NOS3 (0.40) NOS3NOS1NOS2SLC6A2SLC6A4
SCHEMBL8612846 0.87 MRGPRX4 (0.38) HDAC3HDAC1HDAC2NOS3NOS1
SCHEMBL8614188 0.83 MRGPRX4 (0.40) NOS3NOS1NOS2SLC6A2SLC6A4
SCHEMBL9018659 0.81 PLK1 (0.40)
SCHEMBL8612829 0.80 CFTR (0.46) PPARGNR1H2NR1H3
SCHEMBL9018694 0.78 SLC9A1 (0.44)
SCHEMBL9018732 0.77 FFAR4 (0.40)
SCHEMBL9018672 0.76 PIM1 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0743301-A2 Benzoylguanidines containing fluorine MERCK PATENT GmbH (DE) 1996-11-20 EP disclosed