SCHEMBL9019801

SCHEMBL9019801

COc1nc(N)nc2ncn(COC(COC(C)C)COC(C)C)c12

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 9/20 0.36
CDK1 P06493 7/20 0.34
CCNB1 P14635 7/20 0.34
CCNA2 P20248 7/20 0.34
CDK2 P24941 7/20 0.34
CCNA1 P78396 7/20 0.34
HSP90AA1 P07900 1/20 0.32
HSP90AB1 P08238 1/20 0.32
TLR8 Q9NR97 2/20 0.30
ADORA2A P29274 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9019771 0.91 CDK1 (0.40) TLR7CDK1CCNB1CCNA2CDK2
SCHEMBL9019783 0.88 ADORA2A (0.35) TLR7CDK1CCNB1CCNA2CDK2
SCHEMBL9019778 0.82 TLR7 (0.39) TLR7TLR8
SCHEMBL9019784 0.79 ALDH1A1 (0.36)
SCHEMBL9019744 0.77 ALDH1A1 (0.32)
SCHEMBL9019822 0.75 MEN1 (0.48)
SCHEMBL9019742 0.72 ACHE (0.33)
SCHEMBL7981049 0.71 TLR7 (0.39) TLR7CDK1CCNB1CCNA2CDK2
SCHEMBL9019773 0.71 PDE3A (0.39)
Rociclovir SCHEMBL29573658 0.69 ALDH1A1 (0.49) CDK1CCNB1CDK2HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0452680-B1 Substituted purines, process for their preparation and their use as antiviral agents HOECHST AG (DE) 1996-11-06 EP disclosed
EP-0452680-A1 Substituted purines, process for their preparation and their use as antiviral agents HOECHST AKTIENGESELLSCHAFT (DE) 1991-10-23 EP disclosed