SCHEMBL9020401

SCHEMBL9020401

CC[Si](CC)(CC)OCOB(O)c1cccc2c1Cc1ccccc1-2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
PNMT P11086 1/20 0.37
HTR7 P34969 1/20 0.34
HTR2B P41595 1/20 0.34
DRD2 P14416 1/20 0.33
DRD4 P21917 1/20 0.33
DRD3 P35462 1/20 0.33
GABRP O00591 1/20 0.32
GABRD O14764 1/20 0.32
GABRA1 P14867 1/20 0.32
GABRB1 P18505 1/20 0.32
GABRG2 P18507 1/20 0.32
GABRB3 P28472 1/20 0.32
GABRA5 P31644 1/20 0.32
GABRA3 P34903 1/20 0.32
GABRA2 P47869 1/20 0.32
GABRB2 P47870 1/20 0.32
GABRA4 P48169 1/20 0.32
GABRE P78334 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9020874 0.79 PNMT (0.44) NPC1RAB9APNMTHTR7HTR2B
SCHEMBL9020793 0.77 RAB9A (0.45) NPC1RAB9APNMTHTR7HTR2B
SCHEMBL10033961 0.73 NPC1 (0.50) NPC1RAB9APNMTHTR7HTR2B
SCHEMBL6870022 0.72 PNMT (0.54) NPC1RAB9APNMTHTR7HTR2B
SCHEMBL9020390 0.71 PNMT (0.37) NPC1RAB9APNMTHTR7HTR2B
SCHEMBL6649917 0.68 PNMT (0.38) NPC1RAB9APNMTHTR7HTR2B
SCHEMBL1478686 0.67 PNMT (0.52) NPC1RAB9APNMTHTR7HTR2B
SCHEMBL28589725 0.67 PNMT (0.45) NPC1RAB9APNMTHTR7HTR2B
SCHEMBL18343747 0.67 PNMT (0.45) NPC1RAB9APNMTHTR7HTR2B
SCHEMBL6650610 0.66 PNMT (0.37) NPC1RAB9APNMTHTR7HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0669921-A4 PREPARATION OF 2-ARYL CARBAPENEMS VIA A BORONIC ACID COUPLING REACTION. MERCK & CO INC (US) 1996-02-07 EP disclosed
EP-0669921-A1 PREPARATION OF 2-ARYL CARBAPENEMS VIA A BORONIC ACID COUPLING REACTION MERCK & CO. INC. (US) 1995-09-06 EP disclosed
US-5442057-A Preparation of 2-aryl carbapenems via a boronic acid coupling reaction DECAMP ANN (US) 1995-08-15 US disclosed
US-5338875-A Boron containing intermediates useful in the preparation of carbapenems MERCK & CO., INC. (US) 1994-08-16 US disclosed
WO-1994011372-A1 PREPARATION OF 2-ARYL CARBAPENEMS VIA A BORONIC ACID COUPLING REACTION MERCK & CO., INC. (US) 1994-05-26 WO disclosed