SCHEMBL9020874

SCHEMBL9020874

OCOB(O)c1cccc2c1Cc1ccccc1-2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNMT P11086 1/20 0.44
NPC1 O15118 3/20 0.42
RAB9A P51151 3/20 0.42
HTR7 P34969 1/20 0.37
HTR2B P41595 1/20 0.37
DRD2 P14416 2/20 0.36
DRD4 P21917 2/20 0.36
DRD3 P35462 2/20 0.36
PGR P06401 1/20 0.33
KDM4E B2RXH2 2/20 0.31
ALDH1A1 P00352 2/20 0.31
MAPT P10636 2/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
POLB P06746 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA4 P22748 1/20 0.31
CA6 P23280 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9020793 0.83 RAB9A (0.45) PNMTNPC1RAB9AHTR7HTR2B
SCHEMBL9020401 0.79 NPC1 (0.39) PNMTNPC1RAB9AHTR7HTR2B
SCHEMBL10033961 0.79 NPC1 (0.50) PNMTNPC1RAB9AHTR7HTR2B
SCHEMBL1478686 0.75 PNMT (0.52) PNMTNPC1RAB9AHTR7HTR2B
SCHEMBL18343747 0.71 PNMT (0.45) PNMTNPC1RAB9AHTR7HTR2B
Boric Acid SCHEMBL28830312 0.70 PNMT (0.47) PNMTNPC1RAB9AHTR7HTR2B
SCHEMBL30103334 0.70 PNMT (0.63) PNMTNPC1RAB9AHTR7HTR2B
SCHEMBL524602 0.70 PNMT (0.63) PNMTNPC1RAB9AHTR7HTR2B
SCHEMBL263230 0.68 PNMT (0.68) PNMTNPC1RAB9AHTR7HTR2B
SCHEMBL2877998 0.68 PNMT (0.61) PNMTNPC1RAB9AHTR7HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0669921-A4 PREPARATION OF 2-ARYL CARBAPENEMS VIA A BORONIC ACID COUPLING REACTION. MERCK & CO INC (US) 1996-02-07 EP disclosed
EP-0669921-A1 PREPARATION OF 2-ARYL CARBAPENEMS VIA A BORONIC ACID COUPLING REACTION MERCK & CO. INC. (US) 1995-09-06 EP disclosed
US-5442057-A Preparation of 2-aryl carbapenems via a boronic acid coupling reaction DECAMP ANN (US) 1995-08-15 US disclosed
US-5338875-A Boron containing intermediates useful in the preparation of carbapenems MERCK & CO., INC. (US) 1994-08-16 US disclosed
WO-1994011372-A1 PREPARATION OF 2-ARYL CARBAPENEMS VIA A BORONIC ACID COUPLING REACTION MERCK & CO., INC. (US) 1994-05-26 WO disclosed