SCHEMBL902064

SCHEMBL902064

Nc1cc(-c2cccnc2)nc(Nc2cnccn2)c1N1CCN(C(=O)O)CC1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 5/20 0.42
HDAC2 Q92769 5/20 0.42
FAAH O00519 1/20 0.42
NPSR1 Q6W5P4 2/20 0.40
USP2 O75604 1/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HTT P42858 1/20 0.40
KMT2A Q03164 1/20 0.40
KARS1 Q15046 6/20 0.39
KIT P10721 1/20 0.39
HDAC3 O15379 1/20 0.38
LMNA P02545 1/20 0.38
SLC6A7 Q99884 1/20 0.37
CYP2C9 P11712 1/20 0.37
GPR6 P46095 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL902044 0.72 KARS1 (0.51) FAAHMEN1ALDH1A1HTTKMT2A
SCHEMBL901876 0.72 KARS1 (0.71) FAAHUSP2TSHRMEN1ALDH1A1
SCHEMBL901752 0.72 KARS1 (0.73) KARS1SLC6A7
SCHEMBL902003 0.72 KARS1 (0.61) FAAHKARS1LMNASLC6A7
SCHEMBL902071 0.69 KARS1 (0.72) KARS1
SCHEMBL902036 0.68 KARS1 (0.81) MEN1HTTKMT2AKARS1LMNA
SCHEMBL1704270 0.68 KARS1 (0.66) FAAHKARS1
SCHEMBL901857 0.68 KARS1 (0.57) KARS1SLC6A7
SCHEMBL902013 0.67 KARS1 (0.58) KARS1
SCHEMBL901988 0.67 KARS1 (0.55) FAAHKARS1SLC6A7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012041476-A1 PYRIDINE AND ISOQUINOLINE DERIVATIVES AS SYK- AND JAK-KINASE INHIBITORS ALMIRALL, S.A. (ES) 2012-04-05 WO disclosed