SCHEMBL9024010

SCHEMBL9024010

O=C1c2c(-c3ccccc3F)noc2CCC1CCCN1CCN(c2cccc(Cl)c2)CC1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.44
HTR7 P34969 4/20 0.43
HTR1A P08908 2/20 0.43
DRD2 P14416 2/20 0.43
DRD4 P21917 1/20 0.43
DRD3 P35462 1/20 0.43
SLC6A2 P23975 1/20 0.42
SLC6A4 P31645 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
HTR2A P28223 1/20 0.42
HTR6 P50406 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9024250 0.99 KCNH2 (0.43) KCNH2HTR7HTR1ADRD2DRD4
SCHEMBL9024282 0.88 HTR7 (0.42) HTR7HTR1ADRD2HTR2A
Hydrochloric Acid SCHEMBL9024511 0.87 HTR7 (0.41) HTR7DRD2DRD4DRD3
SCHEMBL9024561 0.85 HTR1A (0.45) HTR7HTR1ADRD2DRD4DRD3
SCHEMBL9024223 0.84 HTR2C (0.50) HTR7HTR1ADRD2DRD4DRD3
SCHEMBL9688546 0.82 HTR2C (0.56) HTR7HTR1ADRD2DRD4DRD3
Hydrochloric Acid SCHEMBL9023951 0.82 HTR2C (0.55) HTR7HTR1ADRD2DRD4DRD3
SCHEMBL9024541 0.80 HTR1A (0.53) KCNH2HTR7HTR1ADRD2DRD3
Hydrochloric Acid SCHEMBL9024851 0.80 HTR1A (0.52) KCNH2HTR7HTR1ADRD2DRD3
SCHEMBL9024721 0.80 ADRA1A (0.42) HTR7HTR1ADRD2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5114936-A Antipsychotic and analgesic agents HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-05-19 US claimed
EP-0474012-B1 6,7-Dihydro-3-phenyl-1,2-benzisoxazol-4(5H)-ones and -ols, a process for their preparation and their use as medicaments HOECHST ROUSSEL PHARMA (US) 1996-11-27 EP disclosed
US-5256672-A Antipsychotic, analgesic HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-10-26 US disclosed
US-5180834-A Antipsychotic agents HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-01-19 US disclosed
US-5114936-A Antipsychotic and analgesic agents HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-05-19 US disclosed
EP-0474012-A1 6,7-Dihydro-3-phenyl-1,2-benzisoxazol-4(5H)-ones and -ols, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-03-11 EP disclosed