SCHEMBL9024015

SCHEMBL9024015

O=C1COc2ccccc2C(=O)N1CCCCBr

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.42
DRD2 P14416 3/20 0.42
HTR2A P28223 3/20 0.42
HTR7 P34969 1/20 0.41
DRD3 P35462 1/20 0.41
TSHR P16473 2/20 0.40
HDAC3 O15379 1/20 0.40
TUBB4A P04350 1/20 0.40
TUBB P07437 1/20 0.40
TUBA3C P0DPH7 1/20 0.40
HDAC4 P56524 1/20 0.40
TUBA1B P68363 1/20 0.40
TUBA4A P68366 1/20 0.40
TUBB4B P68371 1/20 0.40
TUBB3 Q13509 1/20 0.40
HDAC1 Q13547 1/20 0.40
TUBB2A Q13885 1/20 0.40
TUBB8 Q3ZCM7 1/20 0.40
TUBA3E Q6PEY2 1/20 0.40
TUBA1A Q71U36 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9025337 0.99 TDP1 (0.42) HTR1ADRD2HTR2AHTR7DRD3
SCHEMBL9369776 0.96 TSHR (0.41) HTR1ADRD2HTR2ATSHRMCHR1
SCHEMBL7479707 0.87 TSHR (0.42) HTR1ADRD2HTR2AHTR7DRD3
SCHEMBL1764705 0.82 ALDH1A1 (0.55) HTR1ADRD2HTR2ATSHRL3MBTL1
SCHEMBL9372268 0.81 KMO (0.45) TSHRHDAC3TUBB4ATUBBTUBA3C
SCHEMBL9375461 0.81 TSHR (0.44) TSHRMAPTKMT2A
SCHEMBL9374266 0.80 TSHR (0.43) TSHRMAPTKMT2A
SCHEMBL9373505 0.80 HTR1A (0.69) HTR1ADRD2HTR2AHTR7DRD3
SCHEMBL9025470 0.79 HRH1 (0.52) HTR1ADRD2HTR7DRD3HDAC3
SCHEMBL9381432 0.79 KMT2A (0.62) HTR1ADRD2HTR7DRD3TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0463810-B1 Heterocyclic compound and psychopharmaceutical composition containing same SUNTORY LTD (JP) 1996-01-10 EP disclosed
EP-0376633-B1 Benzoxazepine derivatives SUNTORY LTD (JP) 1994-10-12 EP disclosed
US-5158947-A CONDENSED HETEROCYCLIC COMPOUNDS AND PSYCHOPHARMACEUTICAL COMPOSITION CONTAINING SAME SUNTORY LIMITED (JP) 1992-10-27 US disclosed
EP-0463810-A1 Heterocyclic compound and psychopharmaceutical composition containing same SUNTORY LIMITED (JP) 1992-01-02 EP disclosed
US-5071845-A Psychotropic or anxyiolytic agent SUNTORY LIMITED (JP) 1991-12-10 US disclosed
EP-0376633-A2 Benzoxazepine derivatives SUNTORY LIMITED (JP) 1990-07-04 EP disclosed