SCHEMBL902403

SCHEMBL902403

CS(=O)(=O)c1ccc2nc(-c3ccc(C4=CC=C(C5CCC(CC(=O)O)CC5)CC4)nc3)[nH]c2c1

nearest known ligand 0.57

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 13/20 0.57
KCNH2 Q12809 8/20 0.52
ADORA2A P29274 4/20 0.52
SOAT1 P35610 4/20 0.51
SCD O00767 4/20 0.49
NPBWR1 P48145 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL902702 0.92 DGAT1 (0.47) DGAT1KCNH2ADORA2ASOAT1SCD
SCHEMBL902157 0.86 DGAT1 (0.75) DGAT1KCNH2ADORA2ASOAT1SCD
SCHEMBL902394 0.81 DGAT1 (0.65) DGAT1KCNH2ADORA2ASOAT1SCD
SCHEMBL902577 0.81 DGAT1 (0.53) DGAT1KCNH2ADORA2ASOAT1
SCHEMBL902570 0.78 DGAT1 (0.44) DGAT1KCNH2ADORA2ASOAT1
SCHEMBL10189664 0.78 DGAT1 (0.60) DGAT1KCNH2ADORA2ASOAT1SCD
SCHEMBL901617 0.75 DGAT1 (0.50) DGAT1KCNH2ADORA2ASOAT1
SCHEMBL10189113 0.73 DGAT1 (0.64) DGAT1SOAT1SCDNPBWR1
SCHEMBL10189564 0.72 DGAT1 (0.47) DGAT1KCNH2SOAT1
SCHEMBL902879 0.72 P4HA1 (0.42) DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012044567-A2 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed