SCHEMBL9024554

SCHEMBL9024554

CN(C)CCNc1ccc(N)cc1F

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NCF1 P14598 2/20 0.44
ALDH1A1 P00352 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
PIM1 P11309 1/20 0.41
PIM3 Q86V86 1/20 0.41
PIM2 Q9P1W9 1/20 0.41
HRH3 Q9Y5N1 1/20 0.40
KMT2A Q03164 1/20 0.39
NQO2 P16083 3/20 0.38
NQO1 P15559 1/20 0.38
SLC2A1 P11166 1/20 0.38
CSF1R P07333 2/20 0.37
BRD4 O60885 1/20 0.36
ATAD2 Q6PL18 1/20 0.36
CYP2C19 P33261 1/20 0.36
ADRA2B P18089 1/20 0.36
NOS1 P29475 1/20 0.35
NOS2 P35228 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4727878 0.90 SMN1; SMN2 (0.44) NCF1PIM1PIM3PIM2KMT2A
Hydrochloric Acid SCHEMBL1641765 0.89 SMN1; SMN2 (0.43) NCF1PIM1PIM3PIM2KMT2A
SCHEMBL15585982 0.83 NCF1 (0.47) NCF1ALDH1A1NPSR1HRH3SLC2A1
SCHEMBL6815177 0.81 ALDH1A1 (0.49) NCF1ALDH1A1NPSR1HRH3KMT2A
SCHEMBL14924462 0.81 NCF1 (0.43) NCF1ALDH1A1NPSR1KMT2ANQO2
SCHEMBL23797765 0.81 IDO1 (0.39) ALDH1A1KMT2ANQO2ADRA2B
SCHEMBL23709737 0.80 FERMT2 (0.41) ALDH1A1ADRA2B
SCHEMBL9023734 0.80 POLB (0.43) NCF1ALDH1A1NPSR1HRH3KMT2A
SCHEMBL3927672 0.79 NCF1 (0.43) NCF1ALDH1A1NPSR1HRH3KMT2A
SCHEMBL18403936 0.79 ADRA2B (0.37) ALDH1A1PIM1NQO2ADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108101926-A Pyrimido five-membered heterocycles containing quinolinone, preparation method and applications 郑州大学 2018-06-01 CN disclosed
EP-2585470-B1 NOVEL FUSED PYRIMIDINE DERIVATIVES FOR INHIBITION OF TYROSINE KINASE ACTIVITY HANMI SCIENCE CO LTD (KR) 2017-01-25 EP disclosed
EP-2975042-A1 NOVEL FUSED PYRIMIDINE DERIVATIVES FOR INHIBITION OF TYROSINE KINASE ACTIVITY Boehringer Ingelheim International GmbH (DE) 2016-01-20 EP disclosed
WO-2011162515-A2 NOVEL FUSED PYRIMIDINE DERIVATIVES FOR INHD3ITION OF TYROSINE KINASE ACTIVITY HANMI HOLDINGS CO. , LTD. (KR) 2011-12-29 WO disclosed
EP-0544400-B1 P-Phenylenediamine substituted by a quaternary ammonium group and an electron withdrawing group BRISTOL MYERS SQUIBB CO (US) 1996-03-13 EP disclosed
EP-0544400-A2 P-Phenylenediamine substituted by a quaternary ammonium group and an electron withdrawing group Bristol-Myers Squibb Company (US) 1993-06-02 EP disclosed
US-5198584-A Developers for hair dyes CLAIROL INC. (US) 1993-03-30 US disclosed
US-5139532-A In a tinctorially effective hair dye developer also containing and an adjuvant selected from surfactans, alkalizing agents, thickeners, chealting agents and perfumes CLAIROL, INC. (US) 1992-08-18 US disclosed