SCHEMBL9024873

SCHEMBL9024873

COc1ccc(CC2c3c(cc(OC)c(OC)c3O)CCN2C(=O)CN(C)C)cc1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C19 P33261 1/20 0.52
BCHE P06276 1/20 0.50
ACHE P22303 1/20 0.50
GAA P10253 1/20 0.46
HTT P42858 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
POLB P06746 1/20 0.44
HCRTR1 O43613 1/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
TP53 P04637 2/20 0.43
KCNH2 Q12809 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dimethylamine SCHEMBL9024883 0.85 CYP3A4 (0.56) CYP3A4CYP2D6CYP2C19BCHEACHE
SCHEMBL8982863 0.81 BCHE (0.74) CYP2D6BCHEACHELMNAKCNH2
SCHEMBL9024220 0.80 BCHE (0.54) CYP3A4CYP2D6CYP2C19BCHEACHE
SCHEMBL9427066 0.76 CYP3A4 (0.45) CYP3A4CYP2D6CYP2C19GAAHTT
SCHEMBL9025225 0.76 HCRTR1 (0.51) CYP3A4CYP2D6CYP2C19BCHEACHE
SCHEMBL25728921 0.73 BCHE (0.61) CYP2D6BCHEACHELMNAKCNH2
SCHEMBL4411747 0.73 MTNR1B (0.66) CYP3A4CYP2D6CYP2C19BCHEACHE
SCHEMBL9024153 0.72 MTNR1B (0.56) CYP3A4CYP2D6CYP2C19BCHEACHE
SCHEMBL9025038 0.71 MTNR1B (0.44) CYP3A4CYP2D6CYP2C19BCHEACHE
SCHEMBL9024245 0.71 LMNA (0.52) CYP2D6BCHEACHEHCRTR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0501693-B1 Isoquinoline derivatives BANYU PHARMA CO LTD (JP) 1996-08-28 EP disclosed
US-5362736-A Alkoxy derivatives for cardiovascular disorders BANYU PHARMACEUTICAL CO., LTD. (JP) 1994-11-08 US disclosed
EP-0501693-A1 Isoquinoline derivatives BANYU PHARMACEUTICAL CO., LTD. (JP) 1992-09-02 EP disclosed