SCHEMBL9026192

SCHEMBL9026192

CCC(C)OCCOc1ccnc(CSc2nc3cc(C)c(C)cc3[nH]2)c1C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 6/20 0.49
CYP3A4 P08684 6/20 0.49
CYP2D6 P10635 6/20 0.49
CYP2C9 P11712 6/20 0.49
CYP2C19 P33261 6/20 0.49
NPC1 O15118 4/20 0.49
RAB9A P51151 4/20 0.49
BRS3 P32247 1/20 0.41
HRH4 Q9H3N8 1/20 0.39
ALDH1A1 P00352 2/20 0.36
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36
AR P10275 1/20 0.36
CYP2E1 P05181 5/20 0.35
CYP2C8 P10632 5/20 0.35
CYP2B6 P20813 5/20 0.35
KMT2A Q03164 2/20 0.35
LMNA P02545 2/20 0.35
MAPT P10636 2/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9025896 0.88 CYP2C9 (0.49) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL8551894 0.88 RAB9A (0.65) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL9027024 0.87 CYP2D6 (0.49) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL9025979 0.86 CYP2C9 (0.56) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL8501930 0.83 CYP2C9 (0.53) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL9026197 0.81 CYP1A2 (0.46) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL9027213 0.79 WDR5 (0.33) CYP2C9ALDH1A1KMT2ALMNAMAPT
SCHEMBL9027225 0.79 WDR5 (0.33) CYP2C9ALDH1A1KMT2ALMNAMAPT
SCHEMBL9026970 0.76 CYP1A2 (0.54) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL8552373 0.74 CYP2D6 (0.54) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0295603-B1 Benzimidazol derivatives and therapeutic agent for ulcer comprising the same EISAI CO LTD (JP) 1996-09-18 EP disclosed
EP-0295603-A1 Benzimidazol derivatives and therapeutic agent for ulcer comprising the same Eisai Co., Ltd. (JP) 1988-12-21 EP disclosed