SCHEMBL9027062

SCHEMBL9027062

CCCC[Si](C)(C)OCCc1c(C(C)=O)n[nH]c1C

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 2/20 0.33
PDE4D Q08499 1/20 0.31
TTR P02766 2/20 0.30
ALB P02768 1/20 0.30
CSNK2A2 P19784 1/20 0.30
KDR P35968 1/20 0.30
CSNK2B P67870 1/20 0.30
CSNK2A1 P68400 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9024908 0.77 HCAR2 (0.31) HCAR2
SCHEMBL9025654 0.76 HCAR2 (0.40) HCAR2PDE4D
SCHEMBL9026160 0.72 HCAR2 (0.37) HCAR2PDE4D
SCHEMBL9025697 0.71 KDM4E (0.43) HCAR2
SCHEMBL8536313 0.70 HCAR2 (0.43) HCAR2PDE4D
SCHEMBL9026200 0.70 CHRNB2 (0.38) HCAR2PDE4D
SCHEMBL7814445 0.70 HCAR2 (0.57) HCAR2
SCHEMBL9037584 0.67 HCAR2 (0.36) HCAR2
SCHEMBL9025309 0.67 HCAR2 (0.41) HCAR2
SCHEMBL3829643 0.65 CES2 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0725783-A1 2-(PYRAZOL-3-YL)CARBAPENEM DERIVATIVES SMITHKLINE BEECHAM PLC (GB) 1996-08-14 EP disclosed
WO-1995011905-A1 2-(PYRAZOL-3-YL)CARBAPENEM DERIVATIVES SMITHKLINE BEECHAM PLC (GB) 1995-05-04 WO disclosed