SCHEMBL9028225

SCHEMBL9028225

C=CCc1c(CCC)c(O)cc2c1OC(C)(C)C2

nearest known ligand 0.38

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
DHFR P00374 2/20 0.38
OSBP P22059 1/20 0.32
HTR2A P28223 1/20 0.32
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9028221 0.79 FFAR4 (0.33) DHFROSBPHTR2APOLB
SCHEMBL9028612 0.79 HTR2A (0.34) OSBPHTR2APOLB
SCHEMBL9027401 0.78 CYP26A1 (0.35) DHFR
SCHEMBL9722348 0.77 POLB (0.33) DHFRPOLB
SCHEMBL9028328 0.76 DHFR (0.33) DHFR
SCHEMBL9027689 0.67 KDM4E (0.36)
SCHEMBL9571543 0.67 LMNA (0.32) HTR2APOLB
SCHEMBL7586358 0.67 OSBP (0.31) OSBP
SCHEMBL14283919 0.66 AKT1 (0.46) DHFRHTR2A
SCHEMBL3961440 0.64 KDM4E (0.46) POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0445827-B1 4-Hydroxytetrahydropyran-2-one derivatives useful as cholesterol and lipid reducing agents FUJIREBIO KK (JP) 1996-09-25 EP disclosed
US-5149834-A Anticholesterol agent and enzyme inhibitors, for curing arteriosclerosis FUJIREBIO INC. (JP) 1992-09-22 US disclosed
EP-0445827-A2 4-Hydroxytetrahydropyran-2-one derivatives useful as cholesterol and lipid reducing agents FUJIREBIO INC. (JP) 1991-09-11 EP disclosed