SCHEMBL9028275

SCHEMBL9028275

COc1ccc(C2(CCOS(C)(=O)=O)CCCNC(C(=O)c3cc(OC)c(OC)c(OC)c3)C2)cc1OC

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 2/20 0.39
TSHR P16473 1/20 0.39
HRH1 P35367 5/20 0.38
L3MBTL1 Q9Y468 1/20 0.36
ALDH1A1 P00352 1/20 0.35
HTT P42858 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
LMNA P02545 2/20 0.35
TACR1 P25103 1/20 0.35
G6PD P11413 1/20 0.35
GAA P10253 1/20 0.34
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9027877 0.91 HRH1 (0.40) HRH1TACR1
SCHEMBL9027955 0.86 ALDH1A1 (0.39) CASP1TSHRALDH1A1HTTMEN1
SCHEMBL8448858 0.80 TSHR (0.35) CASP1TSHRHRH1L3MBTL1ALDH1A1
SCHEMBL27412215 0.80 PKM (0.39) HRH1L3MBTL1ALDH1A1HTTMEN1
SCHEMBL9028321 0.80 MAPT (0.39) CASP1TSHRALDH1A1MEN1KMT2A
SCHEMBL27405658 0.80 L3MBTL1 (0.43) HRH1L3MBTL1ALDH1A1MEN1KMT2A
SCHEMBL9028215 0.79 HRH1 (0.46) HRH1ALDH1A1TACR1
SCHEMBL27401370 0.78 L3MBTL1 (0.37) HRH1L3MBTL1ALDH1A1HTTMEN1
SCHEMBL9028269 0.78 MEN1 (0.39) CASP1TSHRALDH1A1MEN1KMT2A
SCHEMBL9028585 0.78 TACR2 (0.45) HRH1ALDH1A1MEN1KMT2ATACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5563133-A NERVOUS SYSTEM DISORDERS ELI LILLY AND COMPANY (US) 1996-10-08 US disclosed
EP-0714891-A1 Heterocyclic tachykinin receptor antagonists ELI LILLY AND COMPANY (US) 1996-06-05 EP disclosed