SCHEMBL9027877

SCHEMBL9027877

COc1cc(C(=O)C2CC(CCOS(C)(=O)=O)(c3ccc(Cl)c(Cl)c3)CCCN2)cc(OC)c1OC

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 6/20 0.40
TACR2 P21452 3/20 0.40
TACR1 P25103 3/20 0.40
TACR3 P29371 1/20 0.40
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9028275 0.91 CASP1 (0.39) HRH1TACR1
SCHEMBL9028585 0.87 TACR2 (0.45) HRH1TACR2TACR1TACR3SLC6A4
SCHEMBL9028256 0.86 TACR2 (0.43) TACR2TACR1TACR3SLC6A4SLC6A3
SCHEMBL9027899 0.83 TACR2 (0.41) HRH1TACR2TACR1TACR3SLC6A4
SCHEMBL8450883 0.80 TACR2 (0.36) HRH1TACR2TACR1TACR3
SCHEMBL9091759 0.80 HRH1 (0.48) HRH1TACR2TACR1TACR3
SCHEMBL6999634 0.79 TACR2 (0.57) HRH1TACR2TACR1TACR3
SCHEMBL9027870 0.78 TACR2 (0.56) HRH1TACR2TACR1TACR3
SCHEMBL27412215 0.78 PKM (0.39) HRH1
SCHEMBL27405658 0.78 L3MBTL1 (0.43) HRH1TACR2TACR1TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5563133-A NERVOUS SYSTEM DISORDERS ELI LILLY AND COMPANY (US) 1996-10-08 US disclosed
EP-0714891-A1 Heterocyclic tachykinin receptor antagonists ELI LILLY AND COMPANY (US) 1996-06-05 EP disclosed