SCHEMBL902869

SCHEMBL902869

N#Cc1ccc2nc(-c3ccc(-c4ccc(C5CCCCC5)cc4)cc3F)[nH]c2n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CAMKK2 Q96RR4 1/20 0.37
CYP3A4 P08684 2/20 0.36
CYP2C9 P11712 1/20 0.36
APP P05067 1/20 0.36
FASN P49327 2/20 0.36
MAP4K4 O95819 3/20 0.34
CSF1R P07333 3/20 0.34
PIM1 P11309 3/20 0.34
CLK2 P49760 3/20 0.34
MAP4K2 Q12851 3/20 0.34
DYRK1A Q13627 3/20 0.34
MINK1 Q8N4C8 3/20 0.34
AURKB Q96GD4 3/20 0.34
MAP4K5 Q9Y4K4 3/20 0.34
CHEK1 O14757 2/20 0.34
INSR P06213 2/20 0.34
IRAK1 P51617 2/20 0.34
CLK4 Q9HAZ1 2/20 0.34
ALK Q9UM73 2/20 0.34
DYRK3 O43781 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10189555 0.73 SCD (0.54) CYP3A4CYP2C9
SCHEMBL902542 0.70 PDE7A (0.37) CYP3A4CYP2C9APPFASNMAP4K4
SCHEMBL902654 0.68 FASN (0.40) FASNCHEK1DGAT1RAF1
SCHEMBL902790 0.68 DGAT1 (0.51) DGAT1
SCHEMBL902210 0.68 PKN1 (0.60) FASNDGAT1RAF1
SCHEMBL19803789 0.68 CYP3A4 (0.52) CYP3A4CYP2C9APP
SCHEMBL11891678 0.68 CYP3A4 (0.52) CYP3A4CYP2C9APPDHODH
SCHEMBL18411545 0.67 CYP3A4 (0.57) CYP3A4CYP2C9APPDHODHRAF1
SCHEMBL20663895 0.67 CYP3A4 (0.51) CYP3A4CYP2C9APPDHODH
SCHEMBL18458513 0.67 CYP3A4 (0.57) CYP3A4CYP2C9APPDHODHRAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012044567-A2 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed