SCHEMBL9029700

SCHEMBL9029700

N=C(N)c1ccc(C(=O)NCc2ccccc2)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TPSAB1 Q15661 1/20 0.71
HDAC6 Q9UBN7 3/20 0.68
HDAC2 Q92769 1/20 0.68
HDAC8 Q9BY41 1/20 0.68
KLKB1 P03952 3/20 0.64
HPGD P15428 1/20 0.64
CA2 P00918 1/20 0.63
F2 P00734 3/20 0.62
LMNA P02545 1/20 0.62
RAB9A P51151 1/20 0.62
HDAC1 Q13547 2/20 0.61
ROCK2 O75116 1/20 0.59
RPS6KA5 O75582 1/20 0.59
MAP4K4 O95819 1/20 0.59
PRKCG P05129 1/20 0.59
PRKACA P17612 1/20 0.59
RPS6KB1 P23443 1/20 0.59
MAPK1 P28482 1/20 0.59
AKT1 P31749 1/20 0.59
GSK3A P49840 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11900090 0.88 HDAC6 (0.85) HDAC6HDAC2HDAC8HPGDCA2
SCHEMBL6140514 0.86 HDAC6 (0.72) HDAC6HDAC2HDAC8HPGDCA2
SCHEMBL457082 0.84 HDAC6 (0.79) HDAC6HDAC2HDAC8HPGDCA2
SCHEMBL9335737 0.83 TPSAB1 (0.67) TPSAB1HDAC6KLKB1CA2F2
SCHEMBL15606136 0.83 EPHX2 (0.76) TPSAB1HDAC6HDAC2HDAC8KLKB1
SCHEMBL6737728 0.83 HDAC6 (0.72) HDAC6HDAC2HDAC8HPGDCA2
SCHEMBL7983825 0.83 TPSAB1 (0.59) TPSAB1HDAC6KLKB1CA2F2
SCHEMBL4747957 0.82 NR1H4 (0.81) HDAC6HDAC2HDAC8HPGDCA2
SCHEMBL6843720 0.82 HDAC6 (0.77) HDAC6HDAC2HDAC8HPGDCA2
Hydrochloric Acid SCHEMBL3757721 0.82 HDAC6 (0.76) HDAC6HDAC2HDAC8HPGDCA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0730590-A1 NOVEL ISOXAZOLINE AND ISOXAZOLE FIBRINOGEN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-09-11 EP disclosed