SCHEMBL9030286

SCHEMBL9030286

N#Cc1ccc(-c2[c]ccc(C(=N)N)c2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.37
MMP3 P08254 1/20 0.37
MYC P01106 2/20 0.34
CASP1 P29466 2/20 0.34
PRMT1 Q99873 2/20 0.34
ALDH1A1 P00352 1/20 0.34
TOP1 P11387 1/20 0.34
HPGD P15428 1/20 0.34
NQO2 P16083 1/20 0.34
CASP7 P55210 1/20 0.34
HSD17B10 Q99714 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
ASIC3 Q9UHC3 1/20 0.34
PARP15 Q460N3 1/20 0.33
PARP10 Q53GL7 1/20 0.33
PARP2 Q9UGN5 1/20 0.33
CARM1 Q86X55 1/20 0.33
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
PRSS1 P07477 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8169108 0.80 LMNA (0.48) CASP1PRMT1ALDH1A1TOP1HPGD
SCHEMBL8169720 0.80 C1S (0.44) CASP1PRMT1ALDH1A1TOP1HPGD
SCHEMBL8174039 0.80 NQO2 (0.43) CASP1PRMT1ALDH1A1TOP1HPGD
SCHEMBL8170510 0.80 NQO2 (0.44) CASP1PRMT1ALDH1A1TOP1HPGD
SCHEMBL9739115 0.77 MMP3 (0.42) MMP3ALDH1A1KIF11
SCHEMBL8176603 0.76 NQO2 (0.48) IDO1CASP1PRMT1ALDH1A1TOP1
SCHEMBL8176121 0.76 HTT (0.39) CASP1PRMT1ALDH1A1TOP1HPGD
SCHEMBL8163067 0.76 PRSS1 (0.54) IDO1NQO2PARP10PARP2PRSS1
SCHEMBL9219029 0.76 MMP3 (0.52) MMP3ALDH1A1KIF11
SCHEMBL8169371 0.74 PLAU (0.38) NQO2PRSS1PRSS2PRSS3PLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0730590-A1 NOVEL ISOXAZOLINE AND ISOXAZOLE FIBRINOGEN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-09-11 EP disclosed