SCHEMBL9739115

SCHEMBL9739115

N#Cc1ccc(-c2[c]ccc(C#N)c2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP3 P08254 1/20 0.42
KIF11 P52732 3/20 0.38
CA12 O43570 2/20 0.37
CA2 P00918 2/20 0.37
CA9 Q16790 2/20 0.37
CYP2A6 P11509 2/20 0.37
ALDH1A1 P00352 1/20 0.37
CA3 P07451 1/20 0.37
CA6 P23280 1/20 0.37
CA14 Q9ULX7 1/20 0.37
CA1 P00915 1/20 0.36
LOXL2 Q9Y4K0 2/20 0.35
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
NOTUM Q6P988 2/20 0.35
CYP11B2 P19099 2/20 0.35
TNKS O95271 1/20 0.35
TSHR P16473 1/20 0.34
GABRA1 P14867 1/20 0.33
GABRG2 P18507 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9634014 0.87 MMP3 (0.52) MMP3CA12CA2CA9CA3
SCHEMBL1978737 0.87 APP (0.41) MMP3CA12CA2CA9ALDH1A1
SCHEMBL15818998 0.87 MAOA (0.39) ALDH1A1MAOAMAOBNOTUMTSHR
SCHEMBL7194431 0.87 ALDH1A1 (0.47) KIF11CYP2A6ALDH1A1MAOAMAOB
SCHEMBL7526479 0.86 TSHR (0.43) ALDH1A1MAOAMAOBTSHRGABRA1
SCHEMBL9219029 0.83 MMP3 (0.52) MMP3KIF11CA12CA2CA9
SCHEMBL15821103 0.83 KIF11 (0.40) MMP3KIF11CA12CA2CA9
SCHEMBL8532130 0.83 CYP2A6 (0.47) MMP3KIF11CYP2A6ALDH1A1LOXL2
SCHEMBL15819790 0.83 KIF11 (0.39) MMP3KIF11MAOAMAOBCYP11B2
SCHEMBL8530661 0.83 THRB (0.41) ALDH1A1MAOAMAOBTSHRPGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2780326-A1 METHOD FOR INHIBITION OF DEUBIQUITINATING ACTIVITY Vivolux Ab (SE) 2014-09-24 EP disclosed
WO-2014100833-A1 BENZAMIDE COMPOUNDS AND RELATED METHODS OF USE NORTHWESTERN UNIVERSITY (US) 2014-06-26 WO disclosed
WO-2013058691-A1 METHOD FOR INHIBITION OF DEUBIQUITINATING ACTIVITY VIVOLUX AB (SE) 2013-04-25 WO disclosed
CN-101768042-A Method for preparing polysubstituted indene skeleton derivative UNIV FUDAN 2010-07-07 CN disclosed
US-5134150-A Administering diaryl-substituted imidazothiazoles; antiarthritic agents SMITHKLINE BEECHAM CORPORATION (US) 1992-07-28 US disclosed