SCHEMBL9032157

SCHEMBL9032157

CCCCn1c(=O)[nH]c(=S)c2[nH]cnc21

nearest known ligand 0.75

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 14/20 0.75
PDE4B Q07343 14/20 0.75
PDE4C Q08493 14/20 0.75
PDE4D Q08499 14/20 0.75
ADORA2A P29274 13/20 0.75
ADORA2B P29275 10/20 0.62
ADORA3 P0DMS8 3/20 0.62
HPGD P15428 1/20 0.62
ADORA1 P30542 1/20 0.62
BLM P54132 1/20 0.62
PDE3A Q14432 1/20 0.62
HSD17B10 Q99714 1/20 0.62
MEN1 O00255 1/20 0.48
ALDH1A1 P00352 1/20 0.48
KMT2A Q03164 1/20 0.48
BRD4 O60885 1/20 0.47
BRD2 P25440 1/20 0.47
BRD3 Q15059 1/20 0.47
BRDT Q58F21 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8124420 0.92 PDE4A (0.74) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL7990332 0.86 PDE4A (0.58) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL7602847 0.86 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9069127 0.85 ADORA2A (0.72) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL1460898 0.81 PDE4A (0.75) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9791629 0.81 PDE4A (0.89) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL8005197 0.81 ADORA2B (0.59) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL11072066 0.80 PDE4A (0.70) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL11080222 0.79 PDE4A (0.68) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL1376703 0.79 ADORA2A (0.59) PDE4APDE4BPDE4CPDE4DADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0417790-B1 S-triazolo[3,4-i]purine derivatives KYOWA HAKKO KOGYO KK (JP) 1996-12-04 EP disclosed
US-5173492-A Bronchodilator agents KYOWA HAKKO KOGYO CO., LTD. (JP) 1992-12-22 US disclosed
EP-0191313-B1 6-THIOXANTHINE DERIVATIVES Euro-Celtique S.A. (LU) 1992-10-28 EP disclosed
CN-1013676-B 6-THIOXANTHINE DERIVATIVES EURO CELTIQUE SA (US) 1991-08-28 CN disclosed
EP-0417790-A2 S-triazolo[3,4-i]purine derivatives KYOWA HAKKO KOGYO CO., LTD. (JP) 1991-03-20 EP disclosed
US-4820709-A 6-thioxanthine derivatives EUROCELTIQUE, S.A. (LU) 1989-04-11 US disclosed
US-4710503-A 6-thioxanthine derivatives EUROCELTIQUE S.A. (LU) 1987-12-01 US disclosed
CN-86101050-A The manufacture method of 6-Thioxanthine derivatives and application thereof 1986-11-12 CN disclosed
EP-0191313-A1 6-Thioxanthine derivatives Euro-Celtique S.A. (LU) 1986-08-20 EP disclosed