SCHEMBL9033366

SCHEMBL9033366

CCC(Br)c1ccc(C(=O)C2CC2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
LMNA P02545 1/20 0.42
TP53 P04637 1/20 0.42
MAPT P10636 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
CYP2D6 P10635 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
HRH2 P25021 2/20 0.39
HRH1 P35367 2/20 0.39
ESR1 P03372 1/20 0.39
HIF1A Q16665 1/20 0.39
SRD5A2 P31213 1/20 0.39
MGLL Q99685 2/20 0.39
CYP2C19 P33261 1/20 0.38
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
HTR2B P41595 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3750287 0.81 NPC1 (0.49) NPC1RAB9AMEN1KMT2ACYP2D6
SCHEMBL2763268 0.81 NPC1 (0.43) NPC1RAB9ALMNATP53MAPT
SCHEMBL2915168 0.80 LMNA (0.46) NPC1RAB9ALMNATP53MAPT
SCHEMBL3901508 0.77 ALDH1A1 (0.50) LMNATP53MAPTKMT2ACYP2D6
SCHEMBL2923177 0.77 MGLL (0.56) NPC1RAB9ALMNAMEN1KMT2A
SCHEMBL13144199 0.75 NPSR1 (0.54) NPC1RAB9ALMNATP53MAPT
SCHEMBL2762912 0.75 NPC1 (0.41) NPC1RAB9ALMNATP53MAPT
SCHEMBL11550836 0.74 NPC1 (0.49) NPC1RAB9AMEN1KMT2ACYP2D6
SCHEMBL13144197 0.74 NPSR1 (0.52) LMNATP53MAPTL3MBTL1MEN1
SCHEMBL27500533 0.73 HRH2 (0.45) NPC1RAB9ALMNATP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705245-A1 NOVEL INTERMEDIATES FOR THE PREPARATION OF ANTIHISTAMINIC 4-DIPHENYLMETHYL/DIPHENYLMETHOXY PIPERIDINE DERIVATIVES MERRELL PHARMACEUTICALS INC. (US) 1996-04-10 EP disclosed
WO-1995000480-A1 NOVEL INTERMEDIATES FOR THE PREPARATION OF ANTIHISTAMINIC 4-DIPHENYLMETHYL/DIPHENYLMETHOXY PIPERIDINE DERIVATIVES MERRELL PHARMACEUTICALS INC. (US) 1995-01-05 WO disclosed