SCHEMBL9033428

SCHEMBL9033428

Nc1ccc([C]=O)c(Br)c1Br

nearest known ligand 0.31

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 1/20 0.31
CA12 O43570 1/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
CA4 P22748 1/20 0.30
CA6 P23280 1/20 0.30
CA5A P35218 1/20 0.30
CA7 P43166 1/20 0.30
CA9 Q16790 1/20 0.30
CA14 Q9ULX7 1/20 0.30
CA5B Q9Y2D0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22366550 0.76 IMPDH2 (0.42) IMPDH2CA12CA1CA2CA4
SCHEMBL9034278 0.71 ALDH1A1 (0.40) IMPDH2
SCHEMBL19259371 0.70 KDM4E (0.45) CA12CA1CA2CA4CA6
SCHEMBL9312521 0.70
SCHEMBL9328431 0.70 KDM4E (0.41)
SCHEMBL10977537 0.66 IMPDH2 (0.37) IMPDH2CA12CA1CA2CA4
SCHEMBL80034 0.66 AXL (0.38) IMPDH2CA12CA1CA2CA4
SCHEMBL21749799 0.65 CD44 (0.34)
SCHEMBL8590439 0.65 IDO1 (0.46)
SCHEMBL9712649 0.65 NCEH1 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0487095-B1 Pyridyl derivatives, medicines containing these compounds and processes for their preparation THOMAE GMBH DR K (DE) 1996-02-28 EP disclosed
US-5286736-A Thromboxane antagonists and thromboxane synthetase inhibitors DR. KARL THOMAE GMBH (DE) 1994-02-15 US disclosed
EP-0487095-A1 Pyridyl derivatives, medicines containing these compounds and processes for their preparation Dr. Karl Thomae GmbH (DE) 1992-05-27 EP disclosed