SCHEMBL9034278

SCHEMBL9034278

Nc1ccc([C]=O)c(Cl)c1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
TDP1 Q9NUW8 2/20 0.40
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.40
THRB P10828 1/20 0.40
APEX1 P27695 1/20 0.40
RECQL P46063 1/20 0.40
RAB9A P51151 1/20 0.40
BLM P54132 1/20 0.40
KMT2A Q03164 1/20 0.40
MCL1 Q07820 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CYP3A4 P08684 3/20 0.32
TSHR P16473 3/20 0.32
ALOX15 P16050 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
IMPDH2 P12268 1/20 0.31
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL103338 0.84
SCHEMBL20567319 0.76 AR (0.42) ALDH1A1TDP1MEN1NPC1POLB
SCHEMBL526351 0.76 ALDH1A1 (0.50) ALDH1A1TDP1MEN1NPC1POLB
SCHEMBL329657 0.75 MAPK1 (0.40) TDP1CYP3A4MAPK1
SCHEMBL9033428 0.71 IMPDH2 (0.31) IMPDH2
SCHEMBL9712590 0.70 AR (0.36) CYP3A4ALOX15
SCHEMBL6146245 0.70 TSHR (0.52) ALDH1A1TDP1MEN1POLBMAPT
SCHEMBL9311176 0.70 CYP3A4 (0.31) TDP1CYP3A4TSHRMAPK1
SCHEMBL104772 0.69 CYP3A4 (0.32) ALDH1A1TDP1MEN1KMT2ACYP3A4
SCHEMBL103590 0.67 MAPK1 (0.30) TDP1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0487095-B1 Pyridyl derivatives, medicines containing these compounds and processes for their preparation THOMAE GMBH DR K (DE) 1996-02-28 EP disclosed
US-5286736-A Thromboxane antagonists and thromboxane synthetase inhibitors DR. KARL THOMAE GMBH (DE) 1994-02-15 US disclosed
EP-0487095-A1 Pyridyl derivatives, medicines containing these compounds and processes for their preparation Dr. Karl Thomae GmbH (DE) 1992-05-27 EP disclosed