SCHEMBL9033570

SCHEMBL9033570

CC(=O)CC(Cl)c1ccc(C(C)CBr)cc1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
STAT3 P40763 1/20 0.38
ACHE P22303 1/20 0.38
TSHR P16473 2/20 0.37
FFAR1 O14842 2/20 0.35
ALDH1A1 P00352 5/20 0.34
TDP1 Q9NUW8 1/20 0.34
NPSR1 Q6W5P4 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MAPT P10636 1/20 0.32
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31
LMNA P02545 1/20 0.30
HTT P42858 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
HPGD P15428 1/20 0.30
BRD4 O60885 1/20 0.30
CYP1A2 P05177 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9033660 0.84 STAT3 (0.39) STAT3ACHETSHRFFAR1ALDH1A1
SCHEMBL8660435 0.82 POLB (0.42) FFAR1ALDH1A1TDP1KDM4EMAPT
SCHEMBL3822853 0.80 CYP1A2 (0.48) ALDH1A1SMN1; SMN2CYP1A2
SCHEMBL4623899 0.78 ESR1 (0.46) TSHRALDH1A1TDP1KDM4EMAPT
SCHEMBL6935978 0.78 STAT3 (0.46) STAT3ACHEFFAR1ALDH1A1TDP1
SCHEMBL5321358 0.78 BRD4 (0.50) TSHRFFAR1LMNABRD4CYP1A2
SCHEMBL9034467 0.77 FAAH (0.41) TSHRALDH1A1ESR1ESR2LMNA
SCHEMBL3700232 0.77 LMNA (0.41) FFAR1ALDH1A1NPSR1MAPTLMNA
SCHEMBL9034681 0.76 FAAH (0.42) TSHRESR1ESR2LMNA
SCHEMBL4729080 0.76 ALDH1A1 (0.50) TSHRALDH1A1KDM4EMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705245-A1 NOVEL INTERMEDIATES FOR THE PREPARATION OF ANTIHISTAMINIC 4-DIPHENYLMETHYL/DIPHENYLMETHOXY PIPERIDINE DERIVATIVES MERRELL PHARMACEUTICALS INC. (US) 1996-04-10 EP disclosed
WO-1995000480-A1 NOVEL INTERMEDIATES FOR THE PREPARATION OF ANTIHISTAMINIC 4-DIPHENYLMETHYL/DIPHENYLMETHOXY PIPERIDINE DERIVATIVES MERRELL PHARMACEUTICALS INC. (US) 1995-01-05 WO disclosed