SCHEMBL9033591

SCHEMBL9033591

COc1ccc(NC2CCN(CCc3c[nH]c4ccccc34)CC2)cc1OC

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.56
DRD3 P35462 3/20 0.56
ADRA2A P08913 1/20 0.54
ADRA2B P18089 1/20 0.54
ADRA2C P18825 1/20 0.54
ADRA1D P25100 1/20 0.54
ADRA1A P35348 1/20 0.54
ADRA1B P35368 1/20 0.54
MAPT P10636 2/20 0.53
HTR2A P28223 1/20 0.52
HTR1A P08908 3/20 0.49
DRD1 P21728 1/20 0.49
DRD4 P21917 1/20 0.49
DRD5 P21918 1/20 0.49
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL708228 0.83 ADRA2A (0.67) DRD2DRD3ADRA2AADRA2BADRA2C
SCHEMBL12653320 0.80 ALDH1A1 (0.67) ALDH1A1
SCHEMBL11545434 0.79 HTR2A (0.67) DRD2DRD3ADRA2AADRA2BADRA2C
SCHEMBL9027195 0.78 SIGMAR1 (0.54) ADRA1DADRA1AADRA1BHTR1AALDH1A1
SCHEMBL5335494 0.77 HTR2A (0.68) DRD2DRD3ADRA2AADRA2BADRA2C
SCHEMBL9671554 0.76 HTR2A (0.54) DRD2DRD3ADRA2AADRA2BADRA2C
SCHEMBL11545316 0.76 DRD2 (0.63) DRD2DRD3ADRA2AADRA2BADRA2C
SCHEMBL11546493 0.76 DRD2 (0.63) DRD2DRD3ADRA2AADRA2BADRA2C
SCHEMBL5339006 0.75 DRD2 (0.75) DRD2DRD3ADRA2AADRA2BADRA2C
SCHEMBL5336211 0.74 HTR2A (0.64) DRD2DRD3ADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0700385-A1 NOVEL COMPOUNDS SMITHKLINE BEECHAM LABORATOIRES PHARMACEUTIQUES (FR) 1996-03-13 EP disclosed
WO-1994027967-A1 NOVEL COMPOUNDS SMITHKLINE BEECHAM LABORATOIRES PHARMACEUTIQUES (FR) 1994-12-08 WO disclosed