SCHEMBL9033661

SCHEMBL9033661

CC(C)(C)OC(=O)N(CCN(Cc1ccccc1)Cc1ccccc1)CC1CCc2ccccc2O1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.40
SIGMAR1 Q99720 2/20 0.40
ADRA2A P08913 1/20 0.40
ADRA2B P18089 1/20 0.40
ADRA2C P18825 1/20 0.40
CA2 P00918 2/20 0.39
AKT1 P31749 2/20 0.38
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
NCOR2 Q9Y618 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
DRD2 P14416 3/20 0.36
DRD4 P21917 3/20 0.36
DRD3 P35462 3/20 0.36
DRD1 P21728 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8879064 0.88 HTR1A (0.46) HTR1ASIGMAR1ADRA2AADRA2BADRA2C
SCHEMBL9033927 0.85 CA2 (0.45) HTR1ASIGMAR1ADRA2AADRA2BADRA2C
SCHEMBL6286856 0.80 HDAC3 (0.40) AKT1HDAC3HDAC1HDAC2NCOR2
SCHEMBL21091993 0.78 NR1D1 (0.39) CA2
SCHEMBL6285735 0.75 BACE1 (0.40) HDAC3HDAC1HDAC2NCOR2
SCHEMBL9034486 0.74 HTR1A (0.36) HTR1ACA2
SCHEMBL9034476 0.74 HTR1A (0.36) HTR1ACA2
SCHEMBL4934556 0.74 CA2 (0.45) HTR1ASIGMAR1ADRA2AADRA2BADRA2C
SCHEMBL8880016 0.73 CA2 (0.50) HTR1ASIGMAR1ADRA2AADRA2BADRA2C
SCHEMBL8045641 0.73 HRH1 (0.38) L3MBTL1ALDH1A1LMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0639192-B1 (BENZODIOXAN, BENZOFURAN OR BENZOPYRAN)-ALKYLAMINO] ALKYL SUBSTITUTED GUANIDINES AS SELECTIVE VASCOCONSTRICTORS JANSSEN PHARMACEUTICA NV (BE) 1996-05-15 EP disclosed
WO-1993017017-A1 [(BENZODIOXAN, BENZOFURAN OR BENZOPYRAN)-ALKYLAMINO] ALKYL SUBSTITUTED GUANIDINES AS SELECTIVE VASCOCONSTRICTORS JANSSEN PHARMACEUTICA N.V. (BE) 1993-09-02 WO disclosed